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Several compounds showed potent inhibitory activity against sensitive and drug\u2010resistant Gram\u2010positive bacteria. The compounds are ineffective against all tested Gram\u2010negative bacteria. The structure of the ester group exerted a profound effect on antibacterial activity. 4,4\u2010Dimethylcyclohexanyl carbamate <jats:bold>6h<\/jats:bold> exhibited the most potent inhibitory activity against the standard and clinically isolated <jats:italic>Staphylococcus aureus<\/jats:italic>, <jats:italic>Staphylococcus epidermidis<\/jats:italic>, and <jats:italic>Enterococcus faecalis<\/jats:italic> (minimum inhibitory concentration\u2009=\u20094\u20138\u2009\u00b5g\/ml) strains. 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