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For inhibition properties of allylic sulfamates, the half maximal inhibitory concentration (IC<jats:sub>50<\/jats:sub>) and inhibition constant (<jats:italic>K<jats:sub>i<\/jats:sub><\/jats:italic>) were calculated for each novel compounds. The allylic sulfamates showed that <jats:italic>K<jats:sub>i<\/jats:sub><\/jats:italic> values are in the range of 187.33\u2013510.31 pM for hCA I, 104.22\u2013290.09 pM against hCA II, and 12.73\u2013103.63 pM against AChE. The results demonstrated that all newly synthesized compounds had shown effective inhibition against hCA I and II isoenzymes and AChE enzyme.<\/jats:p>","DOI":"10.1002\/jbt.22173","type":"journal-article","created":{"date-parts":[[2018,7,5]],"date-time":"2018-07-05T14:31:50Z","timestamp":1530801110000},"update-policy":"https:\/\/doi.org\/10.1002\/crossmark_policy","source":"Crossref","is-referenced-by-count":33,"title":["Intermolecular amination of allylic and benzylic alcohols leads to effective inhibitions of acetylcholinesterase enzyme and carbonic anhydrase I and II isoenzymes"],"prefix":"10.1002","volume":"32","author":[{"given":"Ufuk","family":"Atmaca","sequence":"first","affiliation":[{"name":"Department of Chemistry Faculty of Science Ataturk University  25240 Erzurum\u2010Turkey"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Alper","family":"Y\u0131ld\u0131r\u0131m","sequence":"additional","affiliation":[{"name":"Department of Chemistry Faculty of Science Ataturk University  25240 Erzurum\u2010Turkey"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Parham","family":"Taslimi","sequence":"additional","affiliation":[{"name":"Department of Chemistry Faculty of Science Ataturk University  25240 Erzurum\u2010Turkey"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Seda Tuncel","family":"\u00c7elik","sequence":"additional","affiliation":[{"name":"Department of Chemistry Faculty of Science Ataturk University  25240 Erzurum\u2010Turkey"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"ORCID":"https:\/\/orcid.org\/0000-0001-5993-1668","authenticated-orcid":false,"given":"\u0130lhami","family":"G\u00fcl\u00e7in","sequence":"additional","affiliation":[{"name":"Department of Chemistry Faculty of Science Ataturk University  25240 Erzurum\u2010Turkey"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Claudiu T.","family":"Supuran","sequence":"additional","affiliation":[{"name":"Dipartimento Di ChimicaUgo Schiff Universita DegliStudi Di Firenze  Firenze Italy"},{"name":"Department of Neurofarba Section of Pharmaceutical and Nutriceutical Sciences Universita DegliStudi Di Firenze  Florence Italy"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Murat","family":"\u00c7elik","sequence":"additional","affiliation":[{"name":"Department of Chemistry Faculty of Science Ataturk University  25240 Erzurum\u2010Turkey"}],"role":[{"vocabulary":"crossref","role":"author"}]}],"member":"311","published-online":{"date-parts":[[2018,7,5]]},"reference":[{"key":"e_1_2_8_2_1","doi-asserted-by":"publisher","DOI":"10.1039\/p19750002413"},{"key":"e_1_2_8_3_1","doi-asserted-by":"publisher","DOI":"10.1021\/ja00836a054"},{"key":"e_1_2_8_4_1","doi-asserted-by":"publisher","DOI":"10.1021\/ja900328x"},{"key":"e_1_2_8_5_1","doi-asserted-by":"publisher","DOI":"10.1002\/ejoc.201100054"},{"key":"e_1_2_8_6_1","doi-asserted-by":"publisher","DOI":"10.3390\/molecules190710103"},{"key":"e_1_2_8_7_1","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2012.750311"},{"key":"e_1_2_8_8_1","doi-asserted-by":"publisher","DOI":"10.1002\/ardp.201400257"},{"key":"e_1_2_8_9_1","doi-asserted-by":"publisher","DOI":"10.25135\/rnp.71.17.04.074"},{"key":"e_1_2_8_10_1","doi-asserted-by":"publisher","DOI":"10.25135\/acg.oc.4.16.05.418"},{"key":"e_1_2_8_11_1","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2014.956310"},{"key":"e_1_2_8_12_1","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmc.2015.04.019"},{"key":"e_1_2_8_13_1","first-page":"841","volume":"29","author":"Hisar O.","year":"2005","journal-title":"Turk. 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