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Bristol Myers Squibb discovered a high affinity CGRP receptor antagonist BMS\u2010927711 for the treatment of migraine now FDA approved as Nurtec\u00ae ODT (rimegepant). Dual\u2010labeled [<jats:sup>14<\/jats:sup>C]\u2010BMS\u2010927711 was prepared and used in a human absorption\u2013distribution\u2013metabolism\u2013elimination (ADME) study. A dual\u2010labeled analog of BMS\u2010927711 was required to fully track the compound's metabolic transformation. 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