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Der Schwerpunkt bei biologisch aktiven POMs liegt gegenw\u00e4rtig auf organisch funktionalisierten POMs und POM\u2010basierten Nanokomposit\u2010Strukturen, da diese Hybride eine erh\u00f6hte Aktivit\u00e4t gegen Tumoren aufweisen, bei einer gleichzeitig deutlich verringerten Toxizit\u00e4t gegen normale Zellen. W\u00e4hrend die Antitumoraktivit\u00e4t von POMs ausreichend beschrieben ist, sind ihre Wirkungsmechanismen noch weitgehend unbekannt. Dieser Aufsatz gibt einen \u00dcberblick \u00fcber die zytotoxischen Effekte von POMs, wobei der Schwerpunkt auf POM\u2010basierten Hybriden und Nanokomposit\u2010Strukturen liegen soll. Postulierte Wirkungsmechanismen werden vorgestellt und molekulare Targets identifiziert. 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