{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2026,5,11]],"date-time":"2026-05-11T23:29:12Z","timestamp":1778542152046,"version":"3.51.4"},"reference-count":29,"publisher":"Springer Science and Business Media LLC","issue":"7","license":[{"start":{"date-parts":[[2011,6,10]],"date-time":"2011-06-10T00:00:00Z","timestamp":1307664000000},"content-version":"tdm","delay-in-days":0,"URL":"http:\/\/www.springer.com\/tdm"}],"content-domain":{"domain":[],"crossmark-restriction":false},"short-container-title":["J Comput Aided Mol Des"],"published-print":{"date-parts":[[2011,7]]},"DOI":"10.1007\/s10822-011-9439-8","type":"journal-article","created":{"date-parts":[[2011,6,9]],"date-time":"2011-06-09T16:42:05Z","timestamp":1307637725000},"page":"669-676","source":"Crossref","is-referenced-by-count":133,"title":["Biosensor-based small molecule fragment screening with biolayer interferometry"],"prefix":"10.1007","volume":"25","author":[{"given":"Charles A.","family":"Wartchow","sequence":"first","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Frank","family":"Podlaski","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Shirley","family":"Li","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Karen","family":"Rowan","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Xiaolei","family":"Zhang","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"David","family":"Mark","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Kuo-Sen","family":"Huang","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]}],"member":"297","published-online":{"date-parts":[[2011,6,10]]},"reference":[{"key":"9439_CR1","volume-title":"Methods in enzymology, 493, fragment-based drug design- tools, practical approaches, and examples","author":"M Congreve","year":"2011","unstructured":"Congreve M, Rich R, Myszka D, Figaroa F, Siegal G, Marshall F (2011) In: Kuo L (ed) Methods in enzymology, 493, fragment-based drug design- tools, practical approaches, and examples. Elsevier, Amsterdam"},{"key":"9439_CR2","unstructured":"Giannetti M (2011) In: Kuo L (ed) Methods in enzymology, 493, fragment-based drug design- tools, practical approaches, and examples. Elsevier, Amsterdam"},{"key":"9439_CR3","doi-asserted-by":"crossref","first-page":"699","DOI":"10.1021\/jm1010513","volume":"54","author":"M Geitmann","year":"2011","unstructured":"Geitmann M, Elinder M, Seeger C, Brandt P, de Esch IJP, Danielson UH (2011) J Med Chem 54:699\u2013708","journal-title":"J Med Chem"},{"key":"9439_CR4","doi-asserted-by":"crossref","first-page":"44","DOI":"10.1021\/ml900002k","volume":"1","author":"I Navratilova","year":"2010","unstructured":"Navratilova I, Hopkins AL (2010) ACS Med Chem Lett 1:44\u201348","journal-title":"ACS Med Chem Lett"},{"issue":"4","key":"9439_CR5","doi-asserted-by":"crossref","first-page":"337","DOI":"10.1177\/1087057109332595","volume":"14","author":"S Perspicace","year":"2009","unstructured":"Perspicace S, Banner D, Benz J, M\u00fcller F, Schlatter D, Huber W (2009) J Biomol Screen 14(4):337\u2013349","journal-title":"J Biomol Screen"},{"key":"9439_CR6","doi-asserted-by":"crossref","first-page":"2990","DOI":"10.1016\/j.bmcl.2008.03.056","volume":"18","author":"SS Antonysamy","year":"2008","unstructured":"Antonysamy SS, Aubol B, Blaney J, Browner MF, Giannetti AM, Harris SF, H\u00e9bert N, Hendle J, Hopkins S, Jefferson E, Kisinger C, Leveque V, Marciano D, McGee E, N\u00e1jera I, Nolan B, Tomimoto M, Torres E, Wright T (2008) Biorg Med Chem Lett 18:2990\u20132995","journal-title":"Biorg Med Chem Lett"},{"issue":"3","key":"9439_CR7","doi-asserted-by":"crossref","first-page":"202","DOI":"10.1177\/1087057108314651","volume":"13","author":"MD H\u00e4m\u00e4l\u00e4inen","year":"2008","unstructured":"H\u00e4m\u00e4l\u00e4inen MD, Zhukov A, Ivarsson M, Fex T, Gottfries J, Karlsson R, Bj\u00f6rsne M (2008) J Biomol Screen 13(3):202\u2013209","journal-title":"J Biomol Screen"},{"key":"9439_CR8","doi-asserted-by":"crossref","first-page":"3449","DOI":"10.1021\/jm8000289","volume":"51","author":"H Nordstr\u00f6m","year":"2008","unstructured":"Nordstr\u00f6m H, Gossas T, H\u00e4m\u00e4l\u00e4inen M, K\u00e4llblad P, Nystr\u00f6m S, Wallberg H, Danielson UH (2008) J Med Chem 51:3449\u20133459","journal-title":"J Med Chem"},{"key":"9439_CR9","doi-asserted-by":"crossref","first-page":"574","DOI":"10.1021\/jm700952v","volume":"51","author":"AM Giannetti","year":"2008","unstructured":"Giannetti AM, Koch BD, Browner MF (2008) J Med Chem 51:574\u2013580","journal-title":"J Med Chem"},{"key":"9439_CR10","doi-asserted-by":"crossref","first-page":"301","DOI":"10.1038\/nrd1343","volume":"3","author":"MR Arkin","year":"2004","unstructured":"Arkin MR, Wells JA (2004) Nat Rev Drug Discov 3:301\u2013317","journal-title":"Nat Rev Drug Discov"},{"key":"9439_CR11","doi-asserted-by":"crossref","first-page":"211","DOI":"10.1038\/nrd2220","volume":"6","author":"PH Hajduk","year":"2007","unstructured":"Hajduk PH, Greer J (2007) Nat Rev Drug Discov 6:211\u2013219","journal-title":"Nat Rev Drug Discov"},{"key":"9439_CR12","doi-asserted-by":"crossref","first-page":"5942","DOI":"10.1021\/jm100059d","volume":"53","author":"CW Murray","year":"2010","unstructured":"Murray CW, Carr MG, Callaghan O, Chessari G, Congreve M, Cowan S, Coyle JE, Downham R, Figueroa E, Frederickson M, Graham B, McMenamin R, O\u2019Brien MA, Patel S, Phillips TR, Williams G, Woodhead AJ, Woolford A (2010) J Med Chem 53:5942\u20135955","journal-title":"J Med Chem"},{"key":"9439_CR13","doi-asserted-by":"crossref","first-page":"2577","DOI":"10.1021\/jm100009z","volume":"53","author":"S Barelier","year":"2010","unstructured":"Barelier S, Pons J, Marcillat O, Lancelin J-M, Krimm I (2010) J Med Chem 53:2577\u20132588","journal-title":"J Med Chem"},{"key":"9439_CR14","unstructured":"Martin E, Wang J, Zaror I, Yu J, Yan K, Doyle M, Feucht P, Shoemaker K, Warne B, Chin M, Blisseth S, Leder L, Meyerhofer M, Wartchow C, Yao D (2011) In: Cooper M (ed) and Mayr LM (co-ed) Label-free technologies for drug discovery. Wiley"},{"key":"9439_CR15","doi-asserted-by":"crossref","first-page":"316","DOI":"10.1016\/j.ab.2004.03.028","volume":"329","author":"DG Myszka","year":"2004","unstructured":"Myszka DG (2004) Anal Biochem 329:316\u2013323","journal-title":"Anal Biochem"},{"key":"9439_CR16","unstructured":"Wartchow C, Yao D, Li P, Heidecker B, Wei J, Choo S, Zuk R (2008) Society for Biochemical sciences annual meeting, St. Louis, Poster P2072"},{"key":"9439_CR17","doi-asserted-by":"crossref","first-page":"94","DOI":"10.1016\/j.ab.2006.08.021","volume":"359","author":"GA Papalia","year":"2006","unstructured":"Papalia GA, Leavitt S, Bynum MA, Katsamba PS, Wilton R, Qiu H, Steukers M, Want S, Bindu L, Phogat S, Giannetti AM, Ryan TE, Pudlak VA, Matusiewicz K, Michelson KM, Nowakowski A, Pham-Baginski A, Brooks J, Tieman BC, Bruce BD, Vaughn M, Baksh M, Cho YH, De Wit M, Smets A, Vandersmissen J, Michiels L, Myszka DG (2006) Anal Biochem 359:94\u2013105","journal-title":"Anal Biochem"},{"key":"9439_CR18","unstructured":"Podlaski F, Wartchow C, Gao L, Li S, Walker S, Ibabecki S, Huang K-S, Mark D (2010) Society for biochemical sciences annual meeting, Phoenix, Poster B209"},{"key":"9439_CR19","unstructured":"Wartchow C, Yao D, Chen J, Ho H, Ikin B, Perillat D, Wicke R, Witte, Zhao L-Z (2010) Society for biochemical sciences annual meeting, Phoenix, Poster B271"},{"key":"9439_CR20","doi-asserted-by":"crossref","first-page":"47","DOI":"10.1038\/nrm2308","volume":"9","author":"RJ Youle","year":"2008","unstructured":"Youle RJ, Strasser A (2008) Nat Rev Mol Cell Biol 9:47\u201359","journal-title":"Nat Rev Mol Cell Biol"},{"key":"9439_CR21","unstructured":"Blagden SP, Willis AE (2011) Nat Rev Clin. Onc advanced on-line publication. doi: 10.1038\/nrclinonc2011.16"},{"key":"9439_CR22","doi-asserted-by":"crossref","first-page":"234","DOI":"10.1021\/cb1002619","volume":"6","author":"KM Comess","year":"2011","unstructured":"Comess KM, Sun C, Abad-Zapatero C, Goedken ER, Gum RJ, Borhani DW, Argiriadi M, Groebe DR, Jia Y, Clampit JE, Haasch DL, Smith HG, Wang S, Song D, Coen ML, Cloutier TE, Tang H, Cheng X, Quinn C, Liu B, Xin Z, Liu G, Fry EH, Stoll V, Ng TI, Banach D, Marcotte D, Burns DJ, Calderwood DJ, Hadjuk PJ (2011) ACS Chem Biol 6:234\u2013244","journal-title":"ACS Chem Biol"},{"issue":"4","key":"9439_CR23","doi-asserted-by":"crossref","first-page":"921","DOI":"10.1110\/ps.8.4.921","volume":"8","author":"D Beckett","year":"1999","unstructured":"Beckett D, Kovaleva E, Schatz J (1999) Prot Sci 8(4):921\u2013929","journal-title":"Prot Sci"},{"key":"9439_CR24","doi-asserted-by":"crossref","first-page":"30","DOI":"10.1016\/j.ab.2010.03.044","volume":"403","author":"G Papalia","year":"2010","unstructured":"Papalia G, Myszka D (2010) Anal Biochem 403:30\u201335","journal-title":"Anal Biochem"},{"key":"9439_CR25","doi-asserted-by":"crossref","first-page":"876","DOI":"10.1038\/nrc1736","volume":"5","author":"SW Fesik","year":"2005","unstructured":"Fesik SW (2005) Nat Rev Cancer 5:876\u2013885","journal-title":"Nat Rev Cancer"},{"issue":"6","key":"9439_CR26","doi-asserted-by":"crossref","first-page":"3012","DOI":"10.1073\/pnas.041619798","volume":"98","author":"AM Petros","year":"2001","unstructured":"Petros AM, Medek A, Nettesheim DG, Kim DH, Yoon HS, Swift K, Matayoshi ED, Oltersdorf T, Fesik SW (2001) PNAS 98(6):3012\u20133017","journal-title":"PNAS"},{"key":"9439_CR27","doi-asserted-by":"crossref","unstructured":"Ku B, Liang C, Jung JU, Oh B-H (2010) Cell Res. doi: 10.1038\/cr.2010.149","DOI":"10.1038\/cr.2010.149"},{"key":"9439_CR28","doi-asserted-by":"crossref","first-page":"615","DOI":"10.1016\/S0022-2836(02)00328-5","volume":"319","author":"A Niedzwieka","year":"2002","unstructured":"Niedzwieka A, Marcotrigiano J, Stepinski J, Jankowska-Anyszka M, Wyslouch-Cieszynska A, Dadlez M, Gingras A-C, Mak P, Darzynkiewicz E, Sonenberg N, Burley SK, Stolarski R (2002) J Mol Biol 319:615\u2013635","journal-title":"J Mol Biol"},{"key":"9439_CR29","doi-asserted-by":"crossref","first-page":"9606","DOI":"10.1021\/ja802977h","volume":"130","author":"KED Coan","year":"2008","unstructured":"Coan KED, Shoichet BK (2008) J Am Chem Soc 130:9606\u20139612","journal-title":"J Am Chem Soc"}],"container-title":["Journal of Computer-Aided Molecular Design"],"original-title":[],"language":"en","link":[{"URL":"http:\/\/link.springer.com\/content\/pdf\/10.1007\/s10822-011-9439-8.pdf","content-type":"application\/pdf","content-version":"vor","intended-application":"text-mining"},{"URL":"http:\/\/link.springer.com\/article\/10.1007\/s10822-011-9439-8\/fulltext.html","content-type":"text\/html","content-version":"vor","intended-application":"text-mining"},{"URL":"http:\/\/link.springer.com\/content\/pdf\/10.1007\/s10822-011-9439-8","content-type":"unspecified","content-version":"vor","intended-application":"similarity-checking"}],"deposited":{"date-parts":[[2019,6,11]],"date-time":"2019-06-11T15:31:13Z","timestamp":1560267073000},"score":1,"resource":{"primary":{"URL":"http:\/\/link.springer.com\/10.1007\/s10822-011-9439-8"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2011,6,10]]},"references-count":29,"journal-issue":{"issue":"7","published-print":{"date-parts":[[2011,7]]}},"alternative-id":["9439"],"URL":"https:\/\/doi.org\/10.1007\/s10822-011-9439-8","relation":{},"ISSN":["0920-654X","1573-4951"],"issn-type":[{"value":"0920-654X","type":"print"},{"value":"1573-4951","type":"electronic"}],"subject":[],"published":{"date-parts":[[2011,6,10]]}}}