{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2026,9,18]],"date-time":"2026-09-18T07:10:48Z","timestamp":1789715448911,"version":"4.0.1"},"reference-count":40,"publisher":"Springer Science and Business Media LLC","issue":"4","license":[{"start":{"date-parts":[[2012,2,1]],"date-time":"2012-02-01T00:00:00Z","timestamp":1328054400000},"content-version":"tdm","delay-in-days":0,"URL":"http:\/\/www.springer.com\/tdm"}],"content-domain":{"domain":[],"crossmark-restriction":false},"short-container-title":["Amino Acids"],"published-print":{"date-parts":[[2012,10]]},"DOI":"10.1007\/s00726-012-1216-z","type":"journal-article","created":{"date-parts":[[2012,1,31]],"date-time":"2012-01-31T12:07:09Z","timestamp":1328011629000},"page":"1431-1443","source":"Crossref","is-referenced-by-count":31,"title":["Site-selective radiolabeling of peptides by 18F-fluorobenzoylation with [18F]SFB in solution and on solid phase: a comparative study"],"prefix":"10.1007","volume":"43","author":[{"given":"Manuela","family":"Kuchar","sequence":"first","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Marc","family":"Pretze","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Torsten","family":"Kniess","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"J\u00f6rg","family":"Steinbach","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Jens","family":"Pietzsch","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Reik","family":"L\u00f6ser","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]}],"member":"297","published-online":{"date-parts":[[2012,2,1]]},"reference":[{"key":"1216_CR1","doi-asserted-by":"crossref","first-page":"243","DOI":"10.2174\/092986706775476070","volume":"13","author":"GD Barry","year":"2006","unstructured":"Barry GD, Le GT, Fairlie DP (2006) Agonists and antagonists of protease activated receptors (PARs). Curr Med Chem 13:243\u2013265","journal-title":"Curr Med Chem"},{"key":"1216_CR2","doi-asserted-by":"crossref","first-page":"2254","DOI":"10.1021\/bc900240z","volume":"20","author":"J Becaud","year":"2009","unstructured":"Becaud J, Mu L, Karramkam M, Schubiger PA, Ametamey SM, Graham K, Stellfeld T, Lehmann L, Borkowski S, Berndorff D, Dinkelborg L, Srinivasan A, Smits R, Koksch B (2009) Direct one-step 18F-labeling of peptides via nucleophilic aromatic substitution. Bioconjugate Chem 20:2254\u20132261","journal-title":"Bioconjugate Chem"},{"key":"1216_CR3","doi-asserted-by":"crossref","first-page":"117","DOI":"10.1002\/jlcr.1826","volume":"54","author":"R Bejot","year":"2011","unstructured":"Bejot R, Elizarov AM, Ball E, Zhang J, Miraghaie R, Kolb HC, Gouverneur V (2011) Batch-mode microfluidic radiosynthesis of N-succinimidyl-4-[18F]fluorobenzoate for protein labelling. J Label Compd Radiopharm 54:117\u2013122","journal-title":"J Label Compd Radiopharm"},{"key":"1216_CR4","doi-asserted-by":"crossref","first-page":"2853","DOI":"10.1002\/ejoc.200800114","volume":"17","author":"LS Cai","year":"2008","unstructured":"Cai LS, Lu SY, Pike VW (2008) Chemistry with [F-18]fluoride ion. Eur J Org Chem 17:2853\u20132873","journal-title":"Eur J Org Chem"},{"key":"1216_CR5","doi-asserted-by":"crossref","first-page":"1005","DOI":"10.1016\/j.addr.2010.09.004","volume":"62","author":"K Chen","year":"2010","unstructured":"Chen K, Conti PS (2010) Target-specific delivery of peptide-based probes for PET imaging. Adv Drug Delivery Rev 62:1005\u20131022","journal-title":"Adv Drug Delivery Rev"},{"key":"1216_CR6","doi-asserted-by":"crossref","first-page":"36505","DOI":"10.1074\/jbc.M706340200","volume":"282","author":"JE Chrencik","year":"2007","unstructured":"Chrencik JE, Brooun A, Recht MI, Nicola G, Davis LK, Abagyan R, Widmer H, Pasquale EB, Kuhn P (2007) Three-dimensional structure of the EphB2 receptor in complex with an antagonistic peptide reveals a novel mode of inhibition. J Biol Chem 282:36505\u201336513","journal-title":"J Biol Chem"},{"key":"1216_CR7","doi-asserted-by":"crossref","first-page":"407","DOI":"10.1002\/jlcr.1656","volume":"52","author":"M Glaser","year":"2009","unstructured":"Glaser M, Robins EG (2009) \u2018Click-labelling\u2019 in PET-radiochemistry. J Label Compd Radiopharm 52:407\u2013414","journal-title":"J Label Compd Radiopharm"},{"key":"1216_CR8","doi-asserted-by":"crossref","first-page":"327","DOI":"10.1002\/jlcr.1601","volume":"52","author":"M Glaser","year":"2009","unstructured":"Glaser M, Arstad E, Luthra SK, Robins EG (2009) Two-step radiosynthesis of [F-18]N-succinimidyl-4-fluorobenzoate ([F-18]SFB). J Label Compd Radiopharm 52:327\u2013330","journal-title":"J Label Compd Radiopharm"},{"key":"1216_CR9","doi-asserted-by":"crossref","first-page":"5901","DOI":"10.1021\/jm800608s","volume":"51","author":"SH Hausner","year":"2008","unstructured":"Hausner SH, Marik J, Gagnon MKJ, Sutcliffe JL (2008) In vivo positron emission tomography (PET) imaging with an \u03b1v\u03b26 specific peptide radiolabeled using 18F-\u201cclick\u201d chemistry: Evaluation and comparison with the corresponding 4-[18F]fluorobenzoyl- and 2-[18F]fluoropropionyl-peptides. J Med Chem 51:5901\u20135904","journal-title":"J Med Chem"},{"key":"1216_CR10","doi-asserted-by":"crossref","first-page":"3005","DOI":"10.1002\/bip.1979.360181208","volume":"18","author":"DL Helseth","year":"1979","unstructured":"Helseth DL, Lechner JH, Veis A (1979) Role of the amino-terminal extra-helical region of type-I collagen in directing the 4D overlap in fibrillogenesis. Biopolymers 18:3005\u20133014","journal-title":"Biopolymers"},{"key":"1216_CR11","volume-title":"Bioconjugate techniques","author":"GT Hermanson","year":"2008","unstructured":"Hermanson GT (2008) Bioconjugate techniques, 2nd edn. Academic Press, Amsterdam","edition":"2"},{"key":"1216_CR12","doi-asserted-by":"crossref","first-page":"143","DOI":"10.1016\/j.pep.2007.10.009","volume":"57","author":"S Hoppmann","year":"2008","unstructured":"Hoppmann S, Haase C, Richter S, Pietzsch J (2008) Expression, purification and fluorine-18 radiolabeling of recombinant S100 proteins\u2014potential probes for molecular imaging of receptor for advanced glycation endproducts (RAGE) in vivo. Protein Expres Purif 57:143\u2013152","journal-title":"Protein Expres Purif"},{"key":"1216_CR13","doi-asserted-by":"crossref","first-page":"422","DOI":"10.1021\/bc100437q","volume":"22","author":"O Jacobson","year":"2011","unstructured":"Jacobson O, Zhu L, Ma Y, Weiss ID, Sun X, Niu G, Kiesewetter DO, Chen X (2011) Rapid and simple one-step F-18 labeling of peptides. Bioconjugate Chem 22:422\u2013428","journal-title":"Bioconjugate Chem"},{"key":"1216_CR14","doi-asserted-by":"crossref","first-page":"595","DOI":"10.1016\/0003-2697(70)90146-6","volume":"34","author":"E Kaiser","year":"1970","unstructured":"Kaiser E, Colescott RL, Bossinger CD, Cook PI (1970) Color test for detection of free terminal amino groups in the solid-phase synthesis of peptides. Anal Biochem 34:595\u2013598","journal-title":"Anal Biochem"},{"key":"1216_CR15","doi-asserted-by":"crossref","first-page":"1218","DOI":"10.1016\/j.apradiso.2011.05.012","volume":"69","author":"J Kapty","year":"2011","unstructured":"Kapty J, Kniess T, Wuest F, Mercer JR (2011) Radiolabeling of phosphatidylserine-binding peptides with prosthetic groups N-[6-(4-[18F]fluorobenzylidene)aminooxyhexyl]maleimide ([18F]FBAM) and N-succinimidyl-4-[18F]fluorobenzoate ([18F]SFB). Appl Radiat Isot 69:1218\u20131225","journal-title":"Appl Radiat Isot"},{"key":"1216_CR16","doi-asserted-by":"crossref","first-page":"255","DOI":"10.1111\/j.1399-3011.1990.tb00976.x","volume":"36","author":"DS King","year":"1990","unstructured":"King DS, Fields CG, Fields GB (1990) A cleavage method which minimizes side reactions following Fmoc solid-phase peptide synthesis. Int J Peptide Protein Res 36:255\u2013266","journal-title":"Int J Peptide Protein Res"},{"key":"1216_CR17","doi-asserted-by":"crossref","first-page":"17301","DOI":"10.1074\/jbc.M500363200","volume":"280","author":"M Koolpe","year":"2005","unstructured":"Koolpe M, Burgess R, Dail M, Pasquale EB (2005) EphB receptor-binding peptides identified by phage display enable design of an antagonist with ephrin-like affinity. J Biol Chem 280:17301\u201317311","journal-title":"J Biol Chem"},{"key":"1216_CR18","doi-asserted-by":"crossref","first-page":"174","DOI":"10.2174\/1874471011003030174","volume":"3","author":"B Kuhnast","year":"2010","unstructured":"Kuhnast B, Dolle F (2010) The challenge of labeling macromolecules with fluorine-18: Three decades of research. Curr Radiopharm 3:174\u2013201","journal-title":"Curr Radiopharm"},{"key":"1216_CR19","doi-asserted-by":"crossref","first-page":"1031","DOI":"10.1016\/j.addr.2010.09.007","volume":"62","author":"Z Li","year":"2010","unstructured":"Li Z, Conti PS (2010) Radiopharmaceutical chemistry for positron emission tomography. Adv Drug Delivery Rev 62:1031\u20131051","journal-title":"Adv Drug Delivery Rev"},{"key":"1216_CR20","doi-asserted-by":"crossref","first-page":"329","DOI":"10.1016\/j.apradiso.2005.03.005","volume":"63","author":"P M\u00e4ding","year":"2005","unstructured":"M\u00e4ding P, F\u00fcchtner F, W\u00fcst F (2005) Module-assisted synthesis of the bifunctional labelling agent N-succinimidyl 4-[F-18]fluorobenzoate ([F-18]SFB). Appl Radiat Isot 63:329\u2013332","journal-title":"Appl Radiat Isot"},{"key":"1216_CR21","doi-asserted-by":"crossref","first-page":"21","DOI":"10.2174\/157019309787316148","volume":"6","author":"C Mamat","year":"2009","unstructured":"Mamat C, Ramenda T, Wuest FR (2009) Recent applications of click chemistry for the synthesis of radiotracers for molecular imaging. Mini-Rev Org Chem 6:21\u201334","journal-title":"Mini-Rev Org Chem"},{"key":"1216_CR22","doi-asserted-by":"crossref","first-page":"1017","DOI":"10.1021\/bc0600564","volume":"17","author":"J Marik","year":"2006","unstructured":"Marik J, Hausner SH, Fix LA, Gagnon MKJ, Sutcliffe JL (2006) Solid-phase synthesis of 2-[18F]fluoropropionyl peptides. Bioconjugate Chem 17:1017\u20131021","journal-title":"Bioconjugate Chem"},{"key":"1216_CR23","doi-asserted-by":"crossref","first-page":"22366","DOI":"10.1016\/S0021-9258(17)31798-2","volume":"269","author":"N Nagan","year":"1994","unstructured":"Nagan N, Kagan HM (1994) Modulation of lysyl oxidase activity toward peptidyl lysine by vicinal dicarboxylic amino acid residues. Implications for collagen cross-linking. J Biol Chem 269:22366\u201322371","journal-title":"J Biol Chem"},{"key":"1216_CR24","doi-asserted-by":"crossref","first-page":"149","DOI":"10.1039\/B922628C","volume":"40","author":"SL Pimlott","year":"2010","unstructured":"Pimlott SL, Sutherland A (2010) Molecular tracers for the PET and SPECT imaging of disease. Chem Soc Rev 40:149\u2013162","journal-title":"Chem Soc Rev"},{"key":"1216_CR25","doi-asserted-by":"crossref","first-page":"241","DOI":"10.1002\/cmdc.200700216","volume":"3","author":"R Rennert","year":"2008","unstructured":"Rennert R, Neundorf I, Jahnke H-G, Suchowerskyj P, Dournaud P, Robitzki A, Beck-Sickinger AG (2008) Generation of carrier peptides for the delivery of nucleic acid drugs in primary cells. ChemMedChem 3:241\u2013253","journal-title":"ChemMedChem"},{"key":"1216_CR26","doi-asserted-by":"crossref","first-page":"479","DOI":"10.1002\/bip.21263","volume":"92","author":"S Richter","year":"2009","unstructured":"Richter S, Bergmann R, Pietzsch J, Ramenda T, Steinbach J, Wuest F (2009) Fluorine-18 labeling of phosphopeptides: A potential approach for the evaluation of phosphopeptide metabolism in vivo. Biopolymers (Pept Sci) 92:479\u2013488","journal-title":"Biopolymers (Pept Sci)"},{"key":"1216_CR27","doi-asserted-by":"crossref","first-page":"243","DOI":"10.2174\/1874471011003030243","volume":"3","author":"TL Ross","year":"2010","unstructured":"Ross TL (2010) The click chemistry approach applied to fluorine-18. Curr Radiopharm 3:243\u2013247","journal-title":"Curr Radiopharm"},{"key":"1216_CR28","first-page":"163","volume-title":"Pharmaceutical radiochemistry (I)","author":"M Schottelius","year":"2010","unstructured":"Schottelius M (2010) Peptide radiopharmaceuticals. In: Wester HJ (ed) Pharmaceutical radiochemistry (I). SCINTOMICS Print Media and Publishing, F\u00fcrstenfeldbruck, pp 163\u2013212"},{"key":"1216_CR29","doi-asserted-by":"crossref","DOI":"10.1002\/352760068X","volume-title":"Peptides: Chemistry and biology","author":"N Sewald","year":"2002","unstructured":"Sewald N, Jakubke H-D (2002) Peptides: Chemistry and biology, 1st edn. Wiley-VCH, Weihnheim","edition":"1"},{"key":"1216_CR30","doi-asserted-by":"crossref","first-page":"2687","DOI":"10.1002\/anie.200352659","volume":"43","author":"NE Shepherd","year":"2004","unstructured":"Shepherd NE, Abbenante G, Fairlie DP (2004) Consecutive cyclic pentapeptide modules form short \u03b1-helices that are very stable to water and denaturants. Angew Chem Int Ed 43:2687\u20132690","journal-title":"Angew Chem Int Ed"},{"key":"1216_CR31","doi-asserted-by":"crossref","first-page":"1501","DOI":"10.1016\/S0960-894X(00)00179-7","volume":"10","author":"JL Sutcliffe-Goulden","year":"2000","unstructured":"Sutcliffe-Goulden JL, O\u2019Doherty MJ, Bansal SS (2000) Solid-phase synthesis of [F-18]labelled peptides for positron emission tomography. Bioorg Med Chem Lett 10:1501\u20131503","journal-title":"Bioorg Med Chem Lett"},{"key":"1216_CR32","doi-asserted-by":"crossref","first-page":"754","DOI":"10.1007\/s00259-001-0756-3","volume":"29","author":"JL Sutcliffe-Goulden","year":"2002","unstructured":"Sutcliffe-Goulden JL, O\u2019Doherty MJ, Marsden PK, Hart IR, Marshall JF, Bansal SS (2002) Rapid solid-phase synthesis and biodistribution of F-18-labelled linear peptides. Eur J Nucl Med Mol Im 29:754\u2013759","journal-title":"Eur J Nucl Med Mol Im"},{"key":"1216_CR33","doi-asserted-by":"crossref","first-page":"68","DOI":"10.1002\/jlcr.1481","volume":"51","author":"G Tang","year":"2008","unstructured":"Tang G, Zeng W, Yu M, Kabalka G (2008) Facile synthesis of N-succinimidyl 4-[18F]fluorobenzoate ([18F]SFB) for protein labeling. J Label Compd Radiopharm 51:68\u201371","journal-title":"J Label Compd Radiopharm"},{"key":"1216_CR34","doi-asserted-by":"crossref","first-page":"543","DOI":"10.1002\/jlcr.1758","volume":"53","author":"GH Tang","year":"2010","unstructured":"Tang GH, Tang XL, Wang XL (2010) A facile automated synthesis of N-succinimidyl 4-[F-18]fluorobenzoate ([F-18]SFB) for F-18-labeled cell-penetrating peptide as PET tracer. J Label Compd Radiopharm 53:543\u2013547","journal-title":"J Label Compd Radiopharm"},{"key":"1216_CR35","doi-asserted-by":"crossref","first-page":"487","DOI":"10.1016\/j.bbagen.2010.02.002","volume":"1800","author":"V Tolmachev","year":"2010","unstructured":"Tolmachev V, Stone-Elander S (2010) Radiolabelled proteins for positron emission tomography: pros and cons of labelling methods. Biochim Biophys Acta 1800:487\u2013510","journal-title":"Biochim Biophys Acta"},{"key":"1216_CR36","doi-asserted-by":"crossref","first-page":"1655","DOI":"10.1038\/nprot.2006.264","volume":"1","author":"G Vaidyanathan","year":"2006","unstructured":"Vaidyanathan G, Zalutsky MR (2006) Synthesis of N-succinimidyl 4-[F-18] fluorobenzoate, an agent for labeling proteins and peptides with F-18. Nat Protoc 1:1655\u20131661","journal-title":"Nat Protoc"},{"key":"1216_CR37","doi-asserted-by":"crossref","first-page":"257","DOI":"10.4155\/fmc.09.28","volume":"1","author":"PM Watt","year":"2009","unstructured":"Watt PM (2009) Phenotypic screening of phylomer peptide libraries derived from genome fragments to identify and validate new targets and therapeutics. Future Med Chem 1:257\u2013265","journal-title":"Future Med Chem"},{"key":"1216_CR38","doi-asserted-by":"crossref","first-page":"79","DOI":"10.1007\/978-3-540-49527-7_4","volume-title":"PET Chemistry: the driving force in molecular imaging","author":"HJ Wester","year":"2007","unstructured":"Wester HJ, Schottelius M (2007) Fluorine-18 labeling of peptides and proteins. In: Schubiger PA, Friebe M, Lehmann L (eds) PET Chemistry: the driving force in molecular imaging. Springer, New York, pp 79\u2013111"},{"key":"1216_CR39","first-page":"S513","volume":"37","author":"HJ Wester","year":"1995","unstructured":"Wester HJ, Krummeich C, Fixmann A, F\u00f6rmer W, M\u00fcller-G\u00e4rtner HW, St\u00f6cklin G (1995) 18F- and 131I-labeling of the octadecapeptide apamin: A selective blocker of the Ca2+ dependent K+-channel. Syntheses and in vivo evaluation in NMRI mice. J Label Compd Radiopharm 37:S513\u2013S515","journal-title":"J Label Compd Radiopharm"},{"key":"1216_CR40","doi-asserted-by":"crossref","first-page":"365","DOI":"10.1016\/0969-8051(96)00017-0","volume":"23","author":"HJ Wester","year":"1996","unstructured":"Wester HJ, Hamacher K, St\u00f6cklin G (1996) A comparative study of NCA fluorine-18 labeling of proteins via acylation and photochemical conjugation. Nucl Med Biol 23:365\u2013372","journal-title":"Nucl Med Biol"}],"container-title":["Amino Acids"],"original-title":[],"language":"en","link":[{"URL":"http:\/\/link.springer.com\/content\/pdf\/10.1007\/s00726-012-1216-z.pdf","content-type":"application\/pdf","content-version":"vor","intended-application":"text-mining"},{"URL":"http:\/\/link.springer.com\/article\/10.1007\/s00726-012-1216-z\/fulltext.html","content-type":"text\/html","content-version":"vor","intended-application":"text-mining"},{"URL":"http:\/\/link.springer.com\/content\/pdf\/10.1007\/s00726-012-1216-z","content-type":"unspecified","content-version":"vor","intended-application":"similarity-checking"}],"deposited":{"date-parts":[[2021,12,27]],"date-time":"2021-12-27T10:51:48Z","timestamp":1640602308000},"score":1,"resource":{"primary":{"URL":"http:\/\/link.springer.com\/10.1007\/s00726-012-1216-z"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2012,2,1]]},"references-count":40,"journal-issue":{"issue":"4","published-print":{"date-parts":[[2012,10]]}},"alternative-id":["1216"],"URL":"https:\/\/doi.org\/10.1007\/s00726-012-1216-z","relation":{},"ISSN":["0939-4451","1438-2199"],"issn-type":[{"value":"0939-4451","type":"print"},{"value":"1438-2199","type":"electronic"}],"subject":[],"published":{"date-parts":[[2012,2,1]]}}}