{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2026,6,11]],"date-time":"2026-06-11T14:24:23Z","timestamp":1781187863878,"version":"3.54.1"},"reference-count":23,"publisher":"Elsevier BV","license":[{"start":{"date-parts":[[2017,4,1]],"date-time":"2017-04-01T00:00:00Z","timestamp":1491004800000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/tdm\/userlicense\/1.0\/"}],"funder":[{"DOI":"10.13039\/501100001824","name":"Czech Science Foundation","doi-asserted-by":"publisher","award":["17-27514Y"],"award-info":[{"award-number":["17-27514Y"]}],"id":[{"id":"10.13039\/501100001824","id-type":"DOI","asserted-by":"publisher"}]},{"DOI":"10.13039\/100007397","name":"Charles University","doi-asserted-by":"publisher","award":["SVV 260 293"],"award-info":[{"award-number":["SVV 260 293"]}],"id":[{"id":"10.13039\/100007397","id-type":"DOI","asserted-by":"publisher"}]},{"name":"University of Pardubice, Faculty of Chemical Technology"}],"content-domain":{"domain":["elsevier.com","sciencedirect.com"],"crossmark-restriction":true},"short-container-title":["Bioorganic Chemistry"],"published-print":{"date-parts":[[2017,4]]},"DOI":"10.1016\/j.bioorg.2017.02.010","type":"journal-article","created":{"date-parts":[[2017,2,21]],"date-time":"2017-02-21T21:00:18Z","timestamp":1487710818000},"page":"244-256","update-policy":"https:\/\/doi.org\/10.1016\/elsevier_cm_policy","source":"Crossref","is-referenced-by-count":9,"special_numbering":"C","title":["Synthesis of readily available fluorophenylalanine derivatives and investigation of their biological activity"],"prefix":"10.1016","volume":"71","author":[{"given":"Martin","family":"Kr\u00e1tk\u00fd","sequence":"first","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"\u0160\u00e1rka","family":"\u0160t\u011bp\u00e1nkov\u00e1","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Katar\u00edna","family":"Vor\u010d\u00e1kov\u00e1","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Lucie","family":"Navr\u00e1tilov\u00e1","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Franti\u0161ek","family":"Trejtnar","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Ji\u0159ina","family":"Stola\u0159\u00edkov\u00e1","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Jarmila","family":"Vin\u0161ov\u00e1","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]}],"member":"78","reference":[{"key":"10.1016\/j.bioorg.2017.02.010_b0005","doi-asserted-by":"crossref","first-page":"203","DOI":"10.1016\/j.jfluchem.2013.09.013","article-title":"N-Hydroxycinnamoyl amides of fluorinated amino acids: synthesis, anti-tyrosinase and DPPH scavenging activities","volume":"156","author":"Chochkova","year":"2013","journal-title":"J. Fluorine Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0010","doi-asserted-by":"crossref","first-page":"5449","DOI":"10.1016\/j.bmcl.2009.07.093","article-title":"Positional effects of monofluorinated phenylalanines on histone acetyltransferase stability and activity","volume":"19","author":"Voloshchuk","year":"2009","journal-title":"Bioorg. Med. Chem. Lett."},{"key":"10.1016\/j.bioorg.2017.02.010_b0015","doi-asserted-by":"crossref","first-page":"2683","DOI":"10.1016\/S0960-894X(01)00542-X","article-title":"Design and synthesis of irreversible depsipeptidyl human rhinovirus 3C protease inhibitors","volume":"11","author":"Webber","year":"2001","journal-title":"Bioorg. Med. Chem. Lett."},{"key":"10.1016\/j.bioorg.2017.02.010_b0020","doi-asserted-by":"crossref","first-page":"494","DOI":"10.1002\/ardp.201100109","article-title":"Design, synthesis, and preliminary activity evaluation of novel peptidomimetics as aminopeptidase N\/CD13 inhibitors","volume":"344","author":"Li","year":"2011","journal-title":"Arch. Pharm. Chem. Life Sci."},{"key":"10.1016\/j.bioorg.2017.02.010_b0025","doi-asserted-by":"crossref","first-page":"1467","DOI":"10.1021\/np070262f","article-title":"Cytotoxic and antihaptotactic beauvericin analogues from precursor-directed biosynthesis with the insect pathogen Beauweria bassiana ATCC 7159","volume":"70","author":"Xu","year":"2007","journal-title":"J. Nat. Prod."},{"key":"10.1016\/j.bioorg.2017.02.010_b0030","doi-asserted-by":"crossref","first-page":"1306","DOI":"10.1016\/j.ejmech.2011.01.053","article-title":"Synthesis and antimycobacterial activity of prodrugs of indeno[2,1-c]quinoline derivatives","volume":"46","author":"Upadhayaya","year":"2011","journal-title":"Eur. J. Med. Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0035","doi-asserted-by":"crossref","first-page":"2061","DOI":"10.1128\/AAC.34.11.2061","article-title":"Action of 1-isonicotinyl-2-palmitoyl hydrazine against the Mycobacterium avium complex and enhancement of its activity by m-fluorophenylalanine","volume":"34","author":"Rastogi","year":"1990","journal-title":"Antimicrob. Agents Chemother."},{"key":"10.1016\/j.bioorg.2017.02.010_b0040","doi-asserted-by":"crossref","first-page":"439","DOI":"10.1021\/jm00287a015","article-title":"Effect of 2-anilinopyridines on protein synthesis","volume":"14","author":"Bailey","year":"1971","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0045","doi-asserted-by":"crossref","first-page":"847","DOI":"10.1002\/ardp.19893221203","article-title":"Investigation on the antiproliferative effects of amino-acid antagonists targeting for aminoacyl-transfer-RNA synthetases. 1. The antibacterial effect","volume":"322","author":"Laske","year":"1989","journal-title":"Arch. Pharm."},{"key":"10.1016\/j.bioorg.2017.02.010_b0050","doi-asserted-by":"crossref","first-page":"5629","DOI":"10.1128\/AAC.00955-13","article-title":"Identification of five structurally unrelated quorum-sensing inhibitors of Pseudomonas aeruginosa from a natural-derivative database","volume":"57","author":"Tan","year":"2013","journal-title":"Antimicrob. Agents Chemother."},{"key":"10.1016\/j.bioorg.2017.02.010_b0055","doi-asserted-by":"crossref","first-page":"904","DOI":"10.1002\/cbdv.201200389","article-title":"Spectroscopically labeled peptaibiotics. Synthesis and properties of selected trichogin GA IV analogs bearing a side-chain-monofluorinated aromatic amino acid for 19F NMR analysis","volume":"10","author":"Peggion","year":"2013","journal-title":"Chem. Biodivers."},{"key":"10.1016\/j.bioorg.2017.02.010_b0060","doi-asserted-by":"crossref","first-page":"1725","DOI":"10.1021\/jm00366a013","article-title":"Transport of antimicrobial agents using peptide carrier systems: anticandidal activity of m-fluorophenylalanine-peptide conjugates","volume":"26","author":"Kingsbury","year":"1983","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0065","doi-asserted-by":"crossref","first-page":"4057","DOI":"10.1128\/AAC.01648-07","article-title":"Enhanced susceptibility to antifungal oligopeptides in yeast strains overexpressing ABC multidrug efflux pumps","volume":"52","author":"Wakiec","year":"2008","journal-title":"Antimicrob. Agents Chemother."},{"key":"10.1016\/j.bioorg.2017.02.010_b0070","doi-asserted-by":"crossref","first-page":"142","DOI":"10.1016\/j.jfluchem.2015.07.006","article-title":"An effective two-step synthesis, fluorescent properties, antioxidant activity and cytotoxicity evaluation of benzene-fluorinated 2,2-dimethyl-2,3-dihydro-1H-quinolin-4-ones","volume":"178","author":"Politanskaya","year":"2015","journal-title":"J. Fluorine Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0075","doi-asserted-by":"crossref","first-page":"4073","DOI":"10.1016\/j.bmc.2014.05.064","article-title":"Synthesis and biological activity of new salicylanilide N,N-disubstituted carbamates and thiocarbamates","volume":"22","author":"Kr\u00e1tk\u00fd","year":"2014","journal-title":"Bioorg. Med. Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0080","doi-asserted-by":"crossref","first-page":"36","DOI":"10.1016\/j.jfluchem.2016.02.004","article-title":"Synthesis and biological activities of novel 1,2,4-triazole thiones and bis(1,2,4-triazole thiones) containing phenylpyrazole and piperazine moieties","volume":"184","author":"Wang","year":"2016","journal-title":"J. Fluorine Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0085","doi-asserted-by":"crossref","first-page":"9426","DOI":"10.3390\/molecules17089426","article-title":"Antifungal activity of salicylanilides and their esters with 4-(trifluoromethyl)benzoic acid","volume":"17","author":"Kr\u00e1tk\u00fd","year":"2012","journal-title":"Molecules"},{"key":"10.1016\/j.bioorg.2017.02.010_b0090","doi-asserted-by":"crossref","first-page":"7453","DOI":"10.1016\/j.bmc.2011.10.042","article-title":"New cholesterol esterase inhibitors based on rhodanine and thiazolidinedione scaffolds","volume":"19","author":"Heng","year":"2011","journal-title":"Bioorg. Med. Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0095","doi-asserted-by":"crossref","first-page":"5213","DOI":"10.1016\/j.bmcl.2008.08.076","article-title":"Tacrine based human cholinesterase inhibitors: synthesis of peptidic-tethered derivatives and their effect on potency and selectivity","volume":"18","author":"Butini","year":"2008","journal-title":"Bioorg. Med. Chem. Lett."},{"key":"10.1016\/j.bioorg.2017.02.010_b0100","doi-asserted-by":"crossref","first-page":"23","DOI":"10.1016\/j.bioorg.2016.07.004","article-title":"Synthesis and in vitro evaluation of novel rhodanine derivatives as potential cholinesterase inhibitors","volume":"68","author":"Kr\u00e1tk\u00fd","year":"2016","journal-title":"Bioorg. Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0105","doi-asserted-by":"crossref","first-page":"106","DOI":"10.1016\/j.bioorg.2015.08.002","article-title":"Synthesis, molecular docking, acetylcholinesterase and butyrylcholinesterase inhibitory potential of thiazole analogs as new inhibitors for Alzheimer disease","volume":"62","author":"Rahim","year":"2015","journal-title":"Bioorg. Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0110","doi-asserted-by":"crossref","first-page":"48","DOI":"10.1016\/j.bioorg.2014.11.005","article-title":"Salicylanilide diethyl phosphates as cholinesterases inhibitors","volume":"58","author":"Kr\u00e1tk\u00fd","year":"2015","journal-title":"Bioorg. Chem."},{"key":"10.1016\/j.bioorg.2017.02.010_b0115","doi-asserted-by":"crossref","first-page":"3674","DOI":"10.3390\/molecules18043674","article-title":"Antibacterial activity of salicylanilide 4-(Trifluoromethyl)-benzoates","volume":"18","author":"Kr\u00e1tk\u00fd","year":"2013","journal-title":"Molecules"}],"container-title":["Bioorganic Chemistry"],"original-title":[],"language":"en","link":[{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0045206816304096?httpAccept=text\/plain","content-type":"text\/plain","content-version":"vor","intended-application":"text-mining"},{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0045206816304096?httpAccept=text\/xml","content-type":"text\/xml","content-version":"vor","intended-application":"text-mining"}],"deposited":{"date-parts":[[2018,9,4]],"date-time":"2018-09-04T00:52:36Z","timestamp":1536022356000},"score":1,"resource":{"primary":{"URL":"https:\/\/linkinghub.elsevier.com\/retrieve\/pii\/S0045206816304096"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2017,4]]},"references-count":23,"alternative-id":["S0045206816304096"],"URL":"https:\/\/doi.org\/10.1016\/j.bioorg.2017.02.010","relation":{},"ISSN":["0045-2068"],"issn-type":[{"value":"0045-2068","type":"print"}],"subject":[],"published":{"date-parts":[[2017,4]]},"assertion":[{"value":"Elsevier","name":"publisher","label":"This article is maintained by"},{"value":"Synthesis of readily available fluorophenylalanine derivatives and investigation of their biological activity","name":"articletitle","label":"Article Title"},{"value":"Bioorganic Chemistry","name":"journaltitle","label":"Journal Title"},{"value":"https:\/\/doi.org\/10.1016\/j.bioorg.2017.02.010","name":"articlelink","label":"CrossRef DOI link to publisher maintained version"},{"value":"article","name":"content_type","label":"Content Type"},{"value":"\u00a9 2017 Elsevier Inc. All rights reserved.","name":"copyright","label":"Copyright"}]}}