{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2026,10,6]],"date-time":"2026-10-06T14:26:01Z","timestamp":1791296761133,"version":"4.1.0"},"reference-count":13,"publisher":"Elsevier BV","issue":"7","license":[{"start":{"date-parts":[[2014,9,1]],"date-time":"2014-09-01T00:00:00Z","timestamp":1409529600000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/tdm\/userlicense\/1.0\/"},{"start":{"date-parts":[[2014,9,1]],"date-time":"2014-09-01T00:00:00Z","timestamp":1409529600000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/legal\/tdmrep-license"}],"funder":[{"name":"Institut F\u00e9d\u00e9ratif de Recherche","award":["IFR 141"],"award-info":[{"award-number":["IFR 141"]}]}],"content-domain":{"domain":["clinicalkey.com","clinicalkey.com.au","clinicalkey.es","clinicalkey.fr","clinicalkey.jp","em-consulte.com","elsevier.com","sciencedirect.com"],"crossmark-restriction":true},"short-container-title":["Biomedicine &amp; Pharmacotherapy"],"published-print":{"date-parts":[[2014,9]]},"DOI":"10.1016\/j.biopha.2014.08.009","type":"journal-article","created":{"date-parts":[[2014,8,19]],"date-time":"2014-08-19T10:15:26Z","timestamp":1408443326000},"page":"893-897","update-policy":"https:\/\/doi.org\/10.1016\/elsevier_cm_policy","source":"Crossref","is-referenced-by-count":13,"title":["Sitamaquine-resistance in Leishmania donovani affects drug accumulation and lipid metabolism"],"prefix":"10.1016","volume":"68","author":[{"given":"L.","family":"Imbert","sequence":"first","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"S.","family":"Cojean","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"D.","family":"Libong","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"P.","family":"Chaminade","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"P.M.","family":"Loiseau","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]}],"member":"78","reference":[{"key":"10.1016\/j.biopha.2014.08.009_bib0005","doi-asserted-by":"crossref","first-page":"1225","DOI":"10.1007\/s00436-011-2555-5","article-title":"Leishmania antimony resistance: what we know what we can learn from the field","volume":"109","author":"A\u00eft-Oudhia","year":"2011","journal-title":"Parasitol Res"},{"key":"10.1016\/j.biopha.2014.08.009_bib0010","doi-asserted-by":"crossref","first-page":"704","DOI":"10.3201\/eid1804.110841","article-title":"Leishmania resistance to miltefosine related to genetic marker","volume":"18","author":"Cojean","year":"2012","journal-title":"Emerg Infect Dis"},{"key":"10.1016\/j.biopha.2014.08.009_bib0015","doi-asserted-by":"crossref","first-page":"246","DOI":"10.1016\/j.bbamem.2006.07.003","article-title":"Interaction of sitamaquine with membrane lipids of Leishmania donovani promastigotes","volume":"1768","author":"Duenas-Romero","year":"2007","journal-title":"Biochim Biophys Acta"},{"key":"10.1016\/j.biopha.2014.08.009_bib0020","doi-asserted-by":"crossref","first-page":"892","DOI":"10.4269\/ajtmh.2011.10-0409","article-title":"Pharmacokinetics of oral sitamaquine taken with or without food and safety and efficacy for treatment of visceral leishmaniasis: a randomized study in Bihar, India","volume":"84","author":"Sundar","year":"2011","journal-title":"Am J Trop Med Hyg"},{"key":"10.1016\/j.biopha.2014.08.009_bib0025","doi-asserted-by":"crossref","first-page":"1425","DOI":"10.1128\/AAC.01123-06","article-title":"Miltefosine affects the lipid metabolism in Leishmania donovani promastigotes","volume":"51","author":"Rakotomanga","year":"2007","journal-title":"Antimicrob Agents Chemother"},{"key":"10.1016\/j.biopha.2014.08.009_bib0030","doi-asserted-by":"crossref","first-page":"164","DOI":"10.1016\/j.biopha.2007.12.006","article-title":"Selection and phenotype characterisation of sitamaquine-resistant promastigotes of Leishmania donovani","volume":"62","author":"Bories","year":"2008","journal-title":"Biomed Pharmacother"},{"key":"10.1016\/j.biopha.2014.08.009_bib0035","doi-asserted-by":"crossref","first-page":"2548","DOI":"10.1093\/jac\/dkq371","article-title":"Mechanism of interaction of sitamaquine with Leishmania donovani","volume":"65","author":"Coimbra","year":"2010","journal-title":"J Antimicrob Chemother"},{"key":"10.1016\/j.biopha.2014.08.009_bib0040","doi-asserted-by":"crossref","first-page":"203","DOI":"10.1016\/S0014-5793(00)01531-3","article-title":"Presence of a Na(+)\/H(+) exchanger in acidocalcisomes of Leishmania donovani and their alkalization by antileishmanial drugs","volume":"473","author":"Vercesi","year":"2000","journal-title":"FEBS Lett"},{"key":"10.1016\/j.biopha.2014.08.009_bib0045","doi-asserted-by":"crossref","first-page":"3838","DOI":"10.1128\/AAC.00065-11","article-title":"Sitamaquine overcomes ABC-mediated resistance to miltefosine and antimony in Leishmania","volume":"55","author":"P\u00e9rez-Victoria","year":"2011","journal-title":"Antimicrob Agents Chemother"},{"key":"10.1016\/j.biopha.2014.08.009_bib0050","doi-asserted-by":"crossref","first-page":"257","DOI":"10.1016\/j.drup.2004.07.002","article-title":"Leishmaniasis: drugs in the clinic, resistance and new developments","volume":"7","author":"Ouellette","year":"2004","journal-title":"Drug Resist Update"},{"key":"10.1016\/j.biopha.2014.08.009_bib0055","doi-asserted-by":"crossref","first-page":"4030","DOI":"10.1128\/AAC.00964-08","article-title":"Sitamaquine sensitivity in Leishmania species is not mediated by drug accumulation in acidocalcisomes","volume":"52","author":"Lopez-Martin","year":"2008","journal-title":"Antimicrob Agents Chemother"},{"key":"10.1016\/j.biopha.2014.08.009_bib0060","first-page":"112","article-title":"Combination therapy with nitazoxanide and amphotericin B, Glucantime\u00ae, miltefosine and sitamaquine against Leishmania (Leishmania) infantum intracellular amastigotes","volume":"130C","author":"Mesquita","year":"2013","journal-title":"Acta Trop"},{"key":"10.1016\/j.biopha.2014.08.009_bib0065","doi-asserted-by":"crossref","first-page":"850","DOI":"10.1093\/jac\/dkq542","article-title":"In vitro interactions between sitamaquine and amphotericin B, sodium stibogluconate, miltefosine, paromomycin and pentamidine against Leishmania donovani","volume":"66","author":"Seifert","year":"2011","journal-title":"J Antimicrobiol Chemother"}],"container-title":["Biomedicine &amp; Pharmacotherapy"],"original-title":[],"language":"en","link":[{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0753332214001036?httpAccept=text\/xml","content-type":"text\/xml","content-version":"vor","intended-application":"text-mining"},{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0753332214001036?httpAccept=text\/plain","content-type":"text\/plain","content-version":"vor","intended-application":"text-mining"}],"deposited":{"date-parts":[[2025,10,10]],"date-time":"2025-10-10T10:54:24Z","timestamp":1760093664000},"score":1,"resource":{"primary":{"URL":"https:\/\/linkinghub.elsevier.com\/retrieve\/pii\/S0753332214001036"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2014,9]]},"references-count":13,"journal-issue":{"issue":"7","published-print":{"date-parts":[[2014,9]]}},"alternative-id":["S0753332214001036"],"URL":"https:\/\/doi.org\/10.1016\/j.biopha.2014.08.009","relation":{},"ISSN":["0753-3322"],"issn-type":[{"value":"0753-3322","type":"print"}],"subject":[],"published":{"date-parts":[[2014,9]]},"assertion":[{"value":"Elsevier","name":"publisher","label":"This article is maintained by"},{"value":"Sitamaquine-resistance in Leishmania donovani affects drug accumulation and lipid metabolism","name":"articletitle","label":"Article Title"},{"value":"Biomedicine & Pharmacotherapy","name":"journaltitle","label":"Journal Title"},{"value":"https:\/\/doi.org\/10.1016\/j.biopha.2014.08.009","name":"articlelink","label":"CrossRef DOI link to publisher maintained version"},{"value":"article","name":"content_type","label":"Content Type"},{"value":"Copyright \u00a9 2014 Elsevier Masson SAS. All rights reserved.","name":"copyright","label":"Copyright"}]}}