{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2025,10,27]],"date-time":"2025-10-27T04:56:32Z","timestamp":1761540992054,"version":"build-2065373602"},"reference-count":27,"publisher":"Elsevier BV","issue":"12","license":[{"start":{"date-parts":[[2010,6,1]],"date-time":"2010-06-01T00:00:00Z","timestamp":1275350400000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/tdm\/userlicense\/1.0\/"},{"start":{"date-parts":[[2010,6,1]],"date-time":"2010-06-01T00:00:00Z","timestamp":1275350400000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/legal\/tdmrep-license"}],"content-domain":{"domain":["elsevier.com","sciencedirect.com"],"crossmark-restriction":true},"short-container-title":["Bioorganic &amp; Medicinal Chemistry"],"published-print":{"date-parts":[[2010,6]]},"DOI":"10.1016\/j.bmc.2010.04.057","type":"journal-article","created":{"date-parts":[[2010,4,26]],"date-time":"2010-04-26T04:47:34Z","timestamp":1272257254000},"page":"4535-4541","update-policy":"https:\/\/doi.org\/10.1016\/elsevier_cm_policy","source":"Crossref","is-referenced-by-count":10,"title":["Development of antiproliferative phenylmaleimides that activate the unfolded protein response"],"prefix":"10.1016","volume":"18","author":[{"given":"Ulrike","family":"Muus","sequence":"first","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Curtis","family":"Hose","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Wei","family":"Yao","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Teresa","family":"Kosakowska-Cholody","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"David","family":"Farnsworth","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Marzena","family":"Dyba","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"George T.","family":"Lountos","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"David S.","family":"Waugh","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Anne","family":"Monks","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"suffix":"Jr.","given":"Terrence R.","family":"Burke","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Christopher J.","family":"Michejda","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]}],"member":"78","reference":[{"key":"10.1016\/j.bmc.2010.04.057_bib1","doi-asserted-by":"crossref","first-page":"1511","DOI":"10.1158\/1535-7163.MCT-05-0485","volume":"5","author":"Kar","year":"2006","journal-title":"Mol. Cancer Ther."},{"key":"10.1016\/j.bmc.2010.04.057_bib2","doi-asserted-by":"crossref","first-page":"33","DOI":"10.1006\/bioo.1996.1052","volume":"25","author":"Ham","year":"1997","journal-title":"Bioorg. Chem."},{"key":"10.1016\/j.bmc.2010.04.057_bib3","doi-asserted-by":"crossref","first-page":"2507","DOI":"10.1016\/S0960-894X(98)00411-9","volume":"8","author":"Ham","year":"1998","journal-title":"Bioorg. Med. Chem. Lett."},{"key":"10.1016\/j.bmc.2010.04.057_bib4","doi-asserted-by":"crossref","first-page":"28304","DOI":"10.1074\/jbc.270.47.28304","volume":"270","author":"Nishikawa","year":"1995","journal-title":"J. Biol. Chem."},{"key":"10.1016\/j.bmc.2010.04.057_bib5","doi-asserted-by":"crossref","first-page":"1217","DOI":"10.1016\/j.bcp.2006.07.024","volume":"72","author":"Kar","year":"2006","journal-title":"Biochem. Pharmacol."},{"key":"10.1016\/j.bmc.2010.04.057_bib6","doi-asserted-by":"crossref","first-page":"2646","DOI":"10.1021\/jo9722055","volume":"63","author":"Choi","year":"1998","journal-title":"J. Org. Chem."},{"key":"10.1016\/j.bmc.2010.04.057_bib7","doi-asserted-by":"crossref","first-page":"185","DOI":"10.1016\/j.ceb.2006.02.003","volume":"18","author":"Boutros","year":"2006","journal-title":"Curr. Opin. Cell Biol."},{"key":"10.1016\/j.bmc.2010.04.057_bib8","doi-asserted-by":"crossref","first-page":"1819","DOI":"10.1093\/clinchem\/48.10.1819","volume":"48","author":"Herzenberg","year":"2002","journal-title":"Clin. Chem."},{"key":"10.1016\/j.bmc.2010.04.057_bib9","doi-asserted-by":"crossref","first-page":"961","DOI":"10.1038\/nrd963","volume":"1","author":"Lyon","year":"2002","journal-title":"Nat. Rev. Drug Disc."},{"key":"10.1016\/j.bmc.2010.04.057_bib10","doi-asserted-by":"crossref","first-page":"880","DOI":"10.1038\/sj.embor.7400779","volume":"7","author":"Szegadi","year":"2006","journal-title":"EMBO Rep."},{"key":"10.1016\/j.bmc.2010.04.057_bib11","doi-asserted-by":"crossref","first-page":"2277","DOI":"10.1089\/ars.2007.1782","volume":"9","author":"Malhotra","year":"2007","journal-title":"Antioxid. Redox Signal."},{"key":"10.1016\/j.bmc.2010.04.057_bib12","doi-asserted-by":"crossref","first-page":"862","DOI":"10.1007\/s00018-007-7383-5","volume":"65","author":"Schr\u00f6der","year":"2008","journal-title":"Cell. Mol. Life Sci."},{"key":"10.1016\/j.bmc.2010.04.057_bib13","doi-asserted-by":"crossref","first-page":"996","DOI":"10.1007\/s10495-009-0341-y","volume":"14","author":"Rasheva","year":"2009","journal-title":"Apoptosis"},{"key":"10.1016\/j.bmc.2010.04.057_bib14","doi-asserted-by":"crossref","first-page":"3604","DOI":"10.1073\/pnas.0510962103","volume":"103","author":"Wang","year":"2006","journal-title":"Proc. Nat. Acad. Sci. U.S.A."},{"key":"10.1016\/j.bmc.2010.04.057_bib15","doi-asserted-by":"crossref","first-page":"519","DOI":"10.1038\/nrm2199","volume":"8","author":"Ron","year":"2007","journal-title":"Nat. Rev. Mol. Cell. Biol."},{"key":"10.1016\/j.bmc.2010.04.057_bib16","doi-asserted-by":"crossref","first-page":"271","DOI":"10.1038\/16729","volume":"397","author":"Harding","year":"1999","journal-title":"Nature"},{"key":"10.1016\/j.bmc.2010.04.057_bib17","doi-asserted-by":"crossref","first-page":"34864","DOI":"10.1074\/jbc.M301107200","volume":"278","author":"Ma","year":"2003","journal-title":"J. Biol. Chem."},{"key":"10.1016\/j.bmc.2010.04.057_bib18","doi-asserted-by":"crossref","first-page":"37375","DOI":"10.1074\/jbc.M303619200","volume":"278","author":"Luo","year":"2003","journal-title":"J. Biol. Chem."},{"key":"10.1016\/j.bmc.2010.04.057_bib19","doi-asserted-by":"crossref","first-page":"S102","DOI":"10.1212\/01.wnl.0000191395.69438.12","volume":"66","author":"Zhang","year":"2006","journal-title":"Neurology"},{"key":"10.1016\/j.bmc.2010.04.057_bib20","doi-asserted-by":"crossref","first-page":"6661","DOI":"10.1074\/jbc.M806735200","volume":"284","author":"Lee","year":"2009","journal-title":"J. Biol. Chem."},{"key":"10.1016\/j.bmc.2010.04.057_bib21","doi-asserted-by":"crossref","first-page":"1011","DOI":"10.1083\/jcb.153.5.1011","volume":"153","author":"Novoa","year":"2001","journal-title":"J. Cell. Biol."},{"key":"10.1016\/j.bmc.2010.04.057_bib22","doi-asserted-by":"crossref","first-page":"3827","DOI":"10.1038\/sj.onc.1206567","volume":"22","author":"Hollander","year":"2003","journal-title":"Oncogene"},{"key":"10.1016\/j.bmc.2010.04.057_bib23","doi-asserted-by":"crossref","first-page":"1242","DOI":"10.1002\/jcb.10711","volume":"90","author":"Yagi","year":"2003","journal-title":"J. Cell. Biochem."},{"key":"10.1016\/j.bmc.2010.04.057_bib24","doi-asserted-by":"crossref","first-page":"716","DOI":"10.1016\/j.semcdb.2007.09.003","volume":"18","author":"Malhotra","year":"2007","journal-title":"Semin. Cell Dev. Biol."},{"key":"10.1016\/j.bmc.2010.04.057_bib25","doi-asserted-by":"crossref","first-page":"1243","DOI":"10.1038\/sj.emboj.7600596","volume":"24","author":"Ohoka","year":"2005","journal-title":"EMBO J."},{"key":"10.1016\/j.bmc.2010.04.057_bib26","doi-asserted-by":"crossref","first-page":"705","DOI":"10.4161\/cbt.6.5.3963","volume":"6","author":"Kadara","year":"2007","journal-title":"Cancer Biol. Ther."},{"key":"10.1016\/j.bmc.2010.04.057_bib27","doi-asserted-by":"crossref","first-page":"1545","DOI":"10.1158\/0008-5472.CAN-08-3858","volume":"69","author":"Schewe","year":"2009","journal-title":"Cancer Res."}],"container-title":["Bioorganic &amp; Medicinal Chemistry"],"original-title":[],"language":"en","link":[{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S096808961000369X?httpAccept=text\/xml","content-type":"text\/xml","content-version":"vor","intended-application":"text-mining"},{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S096808961000369X?httpAccept=text\/plain","content-type":"text\/plain","content-version":"vor","intended-application":"text-mining"}],"deposited":{"date-parts":[[2025,10,18]],"date-time":"2025-10-18T23:46:30Z","timestamp":1760831190000},"score":1,"resource":{"primary":{"URL":"https:\/\/linkinghub.elsevier.com\/retrieve\/pii\/S096808961000369X"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2010,6]]},"references-count":27,"journal-issue":{"issue":"12","published-print":{"date-parts":[[2010,6]]}},"alternative-id":["S096808961000369X"],"URL":"https:\/\/doi.org\/10.1016\/j.bmc.2010.04.057","relation":{},"ISSN":["0968-0896"],"issn-type":[{"type":"print","value":"0968-0896"}],"subject":[],"published":{"date-parts":[[2010,6]]},"assertion":[{"value":"Elsevier","name":"publisher","label":"This article is maintained by"},{"value":"Development of antiproliferative phenylmaleimides that activate the unfolded protein response","name":"articletitle","label":"Article Title"},{"value":"Bioorganic & Medicinal Chemistry","name":"journaltitle","label":"Journal Title"},{"value":"https:\/\/doi.org\/10.1016\/j.bmc.2010.04.057","name":"articlelink","label":"CrossRef DOI link to publisher maintained version"},{"value":"article","name":"content_type","label":"Content Type"},{"value":"Published by Elsevier Ltd.","name":"copyright","label":"Copyright"}]}}