{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2026,9,2]],"date-time":"2026-09-02T06:30:15Z","timestamp":1788330615638,"version":"build-2803163510"},"reference-count":35,"publisher":"Elsevier BV","issue":"7","license":[{"start":{"date-parts":[[2011,4,1]],"date-time":"2011-04-01T00:00:00Z","timestamp":1301616000000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/tdm\/userlicense\/1.0\/"},{"start":{"date-parts":[[2011,4,1]],"date-time":"2011-04-01T00:00:00Z","timestamp":1301616000000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/legal\/tdmrep-license"}],"content-domain":{"domain":["elsevier.com","sciencedirect.com"],"crossmark-restriction":true},"short-container-title":["Bioorganic &amp; Medicinal Chemistry"],"published-print":{"date-parts":[[2011,4]]},"DOI":"10.1016\/j.bmc.2011.02.045","type":"journal-article","created":{"date-parts":[[2011,3,7]],"date-time":"2011-03-07T15:16:18Z","timestamp":1299510978000},"page":"2156-2167","update-policy":"https:\/\/doi.org\/10.1016\/elsevier_cm_policy","source":"Crossref","is-referenced-by-count":35,"title":["Exploration of larger central ring linkers in furamidine analogues: Synthesis and evaluation of their DNA binding, antiparasitic and fluorescence properties"],"prefix":"10.1016","volume":"19","author":[{"given":"Abdelbasset A.","family":"Farahat","sequence":"first","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Ekaterina","family":"Paliakov","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Arvind","family":"Kumar","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Alaa-Eldin M.","family":"Barghash","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Fatma E.","family":"Goda","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Hassan M.","family":"Eisa","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Tanja","family":"Wenzler","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Reto","family":"Brun","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Yang","family":"Liu","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"W. David","family":"Wilson","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"David W.","family":"Boykin","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]}],"member":"78","reference":[{"key":"10.1016\/j.bmc.2011.02.045_b0010","doi-asserted-by":"crossref","first-page":"177","DOI":"10.1080\/00034983.1938.11685024","volume":"32","author":"King","year":"1938","journal-title":"Ann. Trop. Med. Parasitol."},{"key":"10.1016\/j.bmc.2011.02.045_b0015","doi-asserted-by":"crossref","first-page":"289","DOI":"10.1080\/00034983.1939.11685073","volume":"33","author":"Lourie","year":"1939","journal-title":"Ann. Trop. Med. Parasitol."},{"key":"10.1016\/j.bmc.2011.02.045_b0020","first-page":"414","article-title":"Dicationic DNA Minor Groove Binders as Antimicrobial agents","volume":"Vol. 2","author":"Tidwell","year":"2003"},{"key":"10.1016\/j.bmc.2011.02.045_b0025","doi-asserted-by":"crossref","first-page":"232","DOI":"10.1016\/S1471-4922(03)00069-2","volume":"19","author":"Bray","year":"2003","journal-title":"Trends Parasitol."},{"key":"10.1016\/j.bmc.2011.02.045_b0030","doi-asserted-by":"crossref","first-page":"6","DOI":"10.1016\/j.actatropica.2008.07.006","volume":"108","author":"Thuita","year":"2008","journal-title":"Acta Trop."},{"key":"10.1016\/j.bmc.2011.02.045_b0035","doi-asserted-by":"crossref","first-page":"1219","DOI":"10.1021\/jm00219a023","volume":"20","author":"Bijan","year":"1977","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0040","doi-asserted-by":"crossref","first-page":"160","DOI":"10.1002\/jlac.197519750115","volume":"1","author":"Dann","year":"1975","journal-title":"J. Liebigs Ann. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0045","doi-asserted-by":"crossref","first-page":"5324","DOI":"10.1021\/jm060470p","volume":"49","author":"Ismail","year":"2006","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0050","unstructured":"Brun, R.; Werbovetz, K.; Tidwell, R. R.; Boykin, D. W.; Stephens, C. E.; Ismail, M. A.; Kumar, A.; Wilson, W. D. PCT Int. Appl. 2009, p 78. CODEN: PIXXD2 WO 2009051796 A2 20090423 CAN 150:447712 AN 2009:487876."},{"key":"10.1016\/j.bmc.2011.02.045_b0055","doi-asserted-by":"crossref","first-page":"2468","DOI":"10.1021\/jm0612867","volume":"50","author":"Patrick","year":"2007","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0060","doi-asserted-by":"crossref","first-page":"254","DOI":"10.1021\/jm901178d","volume":"53","author":"Bakunov","year":"2010","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0065","doi-asserted-by":"crossref","first-page":"3551","DOI":"10.1016\/j.bmc.2010.03.058","volume":"18","author":"Branowska","year":"2010","journal-title":"Bioorg. Med. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0070","doi-asserted-by":"crossref","first-page":"68","DOI":"10.1002\/jlac.19717490110","volume":"749","author":"Dann","year":"1971","journal-title":"J. Liebigs Ann. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0075","doi-asserted-by":"crossref","first-page":"231","DOI":"10.1128\/AAC.18.2.231","volume":"18","author":"Anne","year":"1980","journal-title":"Antimicrob. Agents Chemother."},{"key":"10.1016\/j.bmc.2011.02.045_b0080","doi-asserted-by":"crossref","first-page":"8452","DOI":"10.1021\/bi00488a036","volume":"29","author":"Wilson","year":"1990","journal-title":"Biochemistry"},{"key":"10.1016\/j.bmc.2011.02.045_b0085","doi-asserted-by":"crossref","first-page":"220","DOI":"10.3109\/10520299509108199","volume":"70","author":"Kapuscinski","year":"1995","journal-title":"Biotech. Histochem."},{"key":"10.1016\/j.bmc.2011.02.045_b0090","doi-asserted-by":"crossref","first-page":"6718","DOI":"10.1016\/j.bmc.2005.07.024","volume":"13","author":"Ismail","year":"2005","journal-title":"Bioorg. Med. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0095","doi-asserted-by":"crossref","first-page":"557","DOI":"10.1016\/j.bmc.2009.12.011","volume":"18","author":"Farahat","year":"2010","journal-title":"Bioorg. Med. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0100","first-page":"707","volume":"5","author":"Kumar","year":"2008","journal-title":"Synthesis"},{"key":"10.1016\/j.bmc.2011.02.045_b0105","series-title":"The Stille Reaction","author":"Farina","year":"1998"},{"key":"10.1016\/j.bmc.2011.02.045_b0110","doi-asserted-by":"crossref","first-page":"2457","DOI":"10.1021\/cr00039a007","volume":"95","author":"Miyaura","year":"1995","journal-title":"Chem. Rev."},{"key":"10.1016\/j.bmc.2011.02.045_b0115","doi-asserted-by":"crossref","first-page":"161","DOI":"10.1016\/0022-328X(87)80017-7","volume":"331","author":"Boere\u2019","year":"1987","journal-title":"J. Organomet. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0120","doi-asserted-by":"crossref","first-page":"4059","DOI":"10.1016\/j.bmcl.2009.06.021","volume":"19","author":"Kuduk","year":"2009","journal-title":"Bioorg. Med. Chem. Lett."},{"key":"10.1016\/j.bmc.2011.02.045_b0125","doi-asserted-by":"crossref","first-page":"4085","DOI":"10.1016\/S0040-4039(03)00834-7","volume":"44","author":"Vyas","year":"2003","journal-title":"Tetrahedron Lett."},{"key":"10.1016\/j.bmc.2011.02.045_b0130","doi-asserted-by":"crossref","first-page":"48","DOI":"10.1246\/cl.2000.48","volume":"1","author":"Sana","year":"2000","journal-title":"Chem. Lett."},{"key":"10.1016\/j.bmc.2011.02.045_b0135","unstructured":"Pasquier, C; Charriere, V; Braun, H. J. Ger. Offen. 2002, DE 10114970; CAN 137: 312310, 202."},{"key":"10.1016\/j.bmc.2011.02.045_b0140","doi-asserted-by":"crossref","first-page":"124","DOI":"10.1021\/jm970570i","volume":"41","author":"Boykin","year":"1998","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0145","doi-asserted-by":"crossref","first-page":"7303","DOI":"10.1016\/S0040-4039(02)01754-9","volume":"43","author":"Seth","year":"2002","journal-title":"Tetrahedron Lett."},{"key":"10.1016\/j.bmc.2011.02.045_b0150","doi-asserted-by":"crossref","first-page":"4330","DOI":"10.1021\/jo040147z","volume":"69","author":"Tao","year":"2004","journal-title":"J. Org. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0155","doi-asserted-by":"crossref","first-page":"999","DOI":"10.1016\/j.biochi.2008.02.017","volume":"90","author":"Wilson","year":"2008","journal-title":"Biochimie"},{"key":"10.1016\/j.bmc.2011.02.045_b0160","doi-asserted-by":"crossref","first-page":"11","DOI":"10.1016\/0301-4622(85)80021-1","volume":"22","author":"Cavatorta","year":"1985","journal-title":"Biophys. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0165","doi-asserted-by":"crossref","first-page":"683","DOI":"10.1016\/j.bmc.2007.10.042","volume":"16","author":"Ismail","year":"2008","journal-title":"Bioorg. Med. Chem."},{"key":"10.1016\/j.bmc.2011.02.045_b0170","doi-asserted-by":"crossref","first-page":"4185","DOI":"10.1128\/AAC.00225-09","volume":"53","author":"Wenzler","year":"2009","journal-title":"Antimicrob. Agents Chemother."},{"key":"10.1016\/j.bmc.2011.02.045_b0175","doi-asserted-by":"crossref","unstructured":"Wilson, W. D.; Tanious, F. A.; Fernandez-Saiz, M.; Rigl, C. T. Evaluation of Drug\u2013Nucleic Acid Interactions by Thermal Melting Curves, In Methods in Molecular Biology, Drug\u2013DNA Interaction Protocols, Fox, K., Ed., 1997; Vol. 90, p 219.","DOI":"10.1385\/0-89603-447-X:219"},{"key":"10.1016\/j.bmc.2011.02.045_b0180","doi-asserted-by":"crossref","first-page":"73","DOI":"10.1016\/0014-5793(95)01537-X","volume":"380","author":"McCoubrey","year":"1996","journal-title":"FEBS Lett."}],"container-title":["Bioorganic &amp; Medicinal Chemistry"],"original-title":[],"language":"en","link":[{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0968089611001635?httpAccept=text\/xml","content-type":"text\/xml","content-version":"vor","intended-application":"text-mining"},{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0968089611001635?httpAccept=text\/plain","content-type":"text\/plain","content-version":"vor","intended-application":"text-mining"}],"deposited":{"date-parts":[[2025,10,18]],"date-time":"2025-10-18T23:53:00Z","timestamp":1760831580000},"score":1,"resource":{"primary":{"URL":"https:\/\/linkinghub.elsevier.com\/retrieve\/pii\/S0968089611001635"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2011,4]]},"references-count":35,"journal-issue":{"issue":"7","published-print":{"date-parts":[[2011,4]]}},"alternative-id":["S0968089611001635"],"URL":"https:\/\/doi.org\/10.1016\/j.bmc.2011.02.045","relation":{},"ISSN":["0968-0896"],"issn-type":[{"value":"0968-0896","type":"print"}],"subject":[],"published":{"date-parts":[[2011,4]]},"assertion":[{"value":"Elsevier","name":"publisher","label":"This article is maintained by"},{"value":"Exploration of larger central ring linkers in furamidine analogues: Synthesis and evaluation of their DNA binding, antiparasitic and fluorescence properties","name":"articletitle","label":"Article Title"},{"value":"Bioorganic & Medicinal Chemistry","name":"journaltitle","label":"Journal Title"},{"value":"https:\/\/doi.org\/10.1016\/j.bmc.2011.02.045","name":"articlelink","label":"CrossRef DOI link to publisher maintained version"},{"value":"article","name":"content_type","label":"Content Type"},{"value":"Copyright \u00a9 2011 Elsevier Ltd. All rights reserved.","name":"copyright","label":"Copyright"}]}}