{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2026,3,6]],"date-time":"2026-03-06T01:54:44Z","timestamp":1772762084354,"version":"3.50.1"},"reference-count":57,"publisher":"Elsevier BV","issue":"2","license":[{"start":{"date-parts":[[2017,1,1]],"date-time":"2017-01-01T00:00:00Z","timestamp":1483228800000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/tdm\/userlicense\/1.0\/"},{"start":{"date-parts":[[2017,1,1]],"date-time":"2017-01-01T00:00:00Z","timestamp":1483228800000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/legal\/tdmrep-license"}],"funder":[{"name":"FP7 European Union","award":["HEALTH-F2-2010-261460"],"award-info":[{"award-number":["HEALTH-F2-2010-261460"]}]},{"name":"DSFP"}],"content-domain":{"domain":["elsevier.com","sciencedirect.com"],"crossmark-restriction":true},"short-container-title":["Bioorganic &amp; Medicinal Chemistry"],"published-print":{"date-parts":[[2017,1]]},"DOI":"10.1016\/j.bmc.2016.11.021","type":"journal-article","created":{"date-parts":[[2016,11,14]],"date-time":"2016-11-14T13:15:46Z","timestamp":1479129346000},"page":"575-580","update-policy":"https:\/\/doi.org\/10.1016\/elsevier_cm_policy","source":"Crossref","is-referenced-by-count":17,"title":["Anion inhibition profiles of the \u03b3-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei responsible of melioidosis and highly drug resistant to common antibiotics"],"prefix":"10.1016","volume":"25","author":[{"given":"Sonia","family":"Del Prete","sequence":"first","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Daniela","family":"Vullo","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Pietro","family":"Di Fonzo","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Sameh M.","family":"Osman","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Zeid","family":"AlOthman","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Claudiu T.","family":"Supuran","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Clemente","family":"Capasso","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]}],"member":"78","reference":[{"key":"10.1016\/j.bmc.2016.11.021_b0005","author":"Miller","year":"2016","journal-title":"Cold Spring Harb Perspect Med"},{"key":"10.1016\/j.bmc.2016.11.021_b0010","doi-asserted-by":"crossref","first-page":"544","DOI":"10.1126\/science.aad9358","volume":"352","author":"Blaser","year":"2016","journal-title":"Science"},{"key":"10.1016\/j.bmc.2016.11.021_b0015","doi-asserted-by":"crossref","first-page":"3","DOI":"10.1016\/j.molcel.2015.10.019","volume":"61","author":"Arenz","year":"2016","journal-title":"Mol Cell"},{"key":"10.1016\/j.bmc.2016.11.021_b0020","doi-asserted-by":"crossref","first-page":"1689","DOI":"10.1517\/14728222.2015.1067685","volume":"19","author":"Capasso","year":"2015","journal-title":"Expert Opin Ther Targets"},{"key":"10.1016\/j.bmc.2016.11.021_b0025","doi-asserted-by":"crossref","first-page":"2130","DOI":"10.2174\/0929867321666141012174921","volume":"22","author":"Capasso","year":"2015","journal-title":"Curr Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0030","doi-asserted-by":"crossref","first-page":"325","DOI":"10.3109\/14756366.2014.910202","volume":"30","author":"Capasso","year":"2015","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0035","doi-asserted-by":"crossref","first-page":"2359","DOI":"10.2174\/1568026616666160413135522","volume":"16","author":"Capasso","year":"2016","journal-title":"Curr Top Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0040","doi-asserted-by":"crossref","first-page":"689","DOI":"10.3109\/14756366.2015.1059333","volume":"31","author":"Ozensoy Guler","year":"2016","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0045","doi-asserted-by":"crossref","first-page":"1254","DOI":"10.1080\/14756366.2016.1201479","volume":"31","author":"Supuran","year":"2016","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0050","doi-asserted-by":"crossref","first-page":"1115","DOI":"10.1016\/j.bmc.2016.01.037","volume":"24","author":"Del Prete","year":"2016","journal-title":"Bioorg Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0055","first-page":"1","author":"Del Prete","year":"2016","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0060","doi-asserted-by":"crossref","first-page":"551","DOI":"10.1517\/14728222.2014.991312","volume":"19","author":"Supuran","year":"2015","journal-title":"Expert Opin Ther Targets"},{"key":"10.1016\/j.bmc.2016.11.021_b0065","doi-asserted-by":"crossref","first-page":"920","DOI":"10.3109\/14756366.2014.990963","volume":"30","author":"Del Prete","year":"2015","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0070","doi-asserted-by":"crossref","first-page":"1385","DOI":"10.1016\/j.bmcl.2015.02.046","volume":"25","author":"De Simone","year":"2015","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0075","doi-asserted-by":"crossref","first-page":"277","DOI":"10.3109\/14756366.2014.917085","volume":"30","author":"De Luca","year":"2015","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0080","doi-asserted-by":"crossref","first-page":"52","DOI":"10.3109\/14756366.2013.877897","volume":"30","author":"Alafeefy","year":"2015","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0085","doi-asserted-by":"crossref","first-page":"9828","DOI":"10.1073\/pnas.1603112113","volume":"113","author":"Kikutani","year":"2016","journal-title":"Proc Natl Acad Sci U S A"},{"key":"10.1016\/j.bmc.2016.11.021_b0090","doi-asserted-by":"crossref","first-page":"4184","DOI":"10.1016\/j.bmcl.2016.07.060","volume":"26","author":"Del Prete","year":"2016","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0095","doi-asserted-by":"crossref","first-page":"4389","DOI":"10.1016\/j.bmcl.2014.08.015","volume":"24","author":"Del Prete","year":"2014","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0100","doi-asserted-by":"crossref","first-page":"1381","DOI":"10.1016\/j.bmcl.2016.01.078","volume":"26","author":"Vullo","year":"2016","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0105","doi-asserted-by":"crossref","first-page":"1156","DOI":"10.3109\/14756366.2015.1102137","volume":"31","author":"Del Prete","year":"2016","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0110","doi-asserted-by":"crossref","first-page":"220","DOI":"10.1016\/j.bmc.2015.12.005","volume":"24","author":"Del Prete","year":"2016","journal-title":"Bioorg Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0115","doi-asserted-by":"crossref","first-page":"810","DOI":"10.3109\/14756366.2015.1069289","volume":"31","author":"De Luca","year":"2016","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0120","doi-asserted-by":"crossref","first-page":"1904","DOI":"10.1002\/cmdc.201600180","volume":"11","author":"Annunziato","year":"2016","journal-title":"ChemMedChem"},{"key":"10.1016\/j.bmc.2016.11.021_b0125","doi-asserted-by":"crossref","first-page":"4537","DOI":"10.1016\/j.bmc.2014.07.048","volume":"22","author":"Prete","year":"2014","journal-title":"Bioorg Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0130","doi-asserted-by":"crossref","first-page":"1127","DOI":"10.1016\/j.bmcl.2013.12.124","volume":"24","author":"Nishimori","year":"2014","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0135","doi-asserted-by":"crossref","first-page":"2939","DOI":"10.1016\/j.bmc.2014.04.006","volume":"22","author":"Nishimori","year":"2014","journal-title":"Bioorg Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0140","doi-asserted-by":"crossref","first-page":"146","DOI":"10.3109\/14756366.2012.761608","volume":"29","author":"Migliardini","year":"2014","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0145","doi-asserted-by":"crossref","first-page":"141","DOI":"10.1016\/j.bmc.2013.11.042","volume":"22","author":"Alafeefy","year":"2014","journal-title":"Bioorg Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0150","doi-asserted-by":"crossref","first-page":"379","DOI":"10.3109\/14756366.2013.787422","volume":"29","author":"Capasso","year":"2014","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0155","doi-asserted-by":"crossref","first-page":"693","DOI":"10.1517\/13543776.2013.778245","volume":"23","author":"Capasso","year":"2013","journal-title":"Expert Opin Ther Pat"},{"key":"10.1016\/j.bmc.2016.11.021_b0160","doi-asserted-by":"crossref","first-page":"144","DOI":"10.59566\/IJBS.2007.3144","volume":"3","author":"Gilad","year":"2007","journal-title":"Int J Biomed Sci"},{"key":"10.1016\/j.bmc.2016.11.021_b0165","doi-asserted-by":"crossref","first-page":"1500","DOI":"10.1097\/CCM.0000000000001668","volume":"44","author":"Stephens","year":"2016","journal-title":"Crit Care Med"},{"key":"10.1016\/j.bmc.2016.11.021_b0170","doi-asserted-by":"crossref","first-page":"169","DOI":"10.1111\/nep.12024","volume":"18","author":"Jabbar","year":"2013","journal-title":"Nephrology (Carlton)"},{"key":"10.1016\/j.bmc.2016.11.021_b0175","doi-asserted-by":"crossref","first-page":"11","DOI":"10.1016\/j.abb.2012.10.010","volume":"529","author":"Zimmerman","year":"2013","journal-title":"Arch Biochem Biophys"},{"key":"10.1016\/j.bmc.2016.11.021_b0180","first-page":"3327","volume":"14","author":"Innocenti","year":"2004","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0185","doi-asserted-by":"crossref","first-page":"9232","DOI":"10.1021\/bi0001877","volume":"39","author":"Tripp","year":"2000","journal-title":"Biochemistry"},{"key":"10.1016\/j.bmc.2016.11.021_b0190","doi-asserted-by":"crossref","first-page":"9222","DOI":"10.1021\/bi000204s","volume":"39","author":"Iverson","year":"2000","journal-title":"Biochemistry"},{"key":"10.1016\/j.bmc.2016.11.021_b0195","doi-asserted-by":"crossref","first-page":"592","DOI":"10.3109\/14756366.2014.957202","volume":"30","author":"Alafeefy","year":"2015","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0200","doi-asserted-by":"crossref","first-page":"240","DOI":"10.1016\/j.bmcl.2013.11.030","volume":"24","author":"Vullo","year":"2014","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0205","doi-asserted-by":"crossref","first-page":"532","DOI":"10.3109\/14756366.2013.822371","volume":"29","author":"Del Prete","year":"2014","journal-title":"J Enzyme Inhib Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0210","doi-asserted-by":"crossref","first-page":"4006","DOI":"10.1016\/j.bmcl.2014.06.024","volume":"24","author":"Ceruso","year":"2014","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0215","doi-asserted-by":"crossref","first-page":"4067","DOI":"10.1016\/j.bmcl.2013.05.063","volume":"23","author":"Del Prete","year":"2013","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0220","doi-asserted-by":"crossref","first-page":"1728","DOI":"10.1016\/j.bmc.2015.02.045","volume":"23","author":"Vullo","year":"2015","journal-title":"Bioorg Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0225","doi-asserted-by":"crossref","first-page":"4970","DOI":"10.1016\/j.bmcl.2015.03.010","volume":"25","author":"De Luca","year":"2015","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0230","doi-asserted-by":"crossref","first-page":"3550","DOI":"10.1016\/j.bmcl.2015.06.079","volume":"25","author":"Vullo","year":"2015","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0235","doi-asserted-by":"crossref","first-page":"4405","DOI":"10.1016\/j.bmc.2015.06.021","volume":"23","author":"De Luca","year":"2015","journal-title":"Bioorg Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0240","doi-asserted-by":"crossref","first-page":"2561","DOI":"10.1016\/S0021-9258(18)62326-9","volume":"246","author":"Khalifah","year":"1971","journal-title":"J Biol Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0245","doi-asserted-by":"crossref","first-page":"1406","DOI":"10.1016\/j.bmcl.2016.01.072","volume":"26","author":"Vullo","year":"2016","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0250","doi-asserted-by":"crossref","first-page":"3413","DOI":"10.1016\/j.bmc.2016.05.029","volume":"24","author":"Del Prete","year":"2016","journal-title":"Bioorg Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0255","doi-asserted-by":"crossref","first-page":"835","DOI":"10.1016\/j.bmc.2016.01.005","volume":"24","author":"De Luca","year":"2016","journal-title":"Bioorg Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0260","doi-asserted-by":"crossref","first-page":"4402","DOI":"10.1016\/j.bmcl.2014.08.014","volume":"24","author":"Vullo","year":"2014","journal-title":"Bioorg Med Chem Lett"},{"key":"10.1016\/j.bmc.2016.11.021_b0265","doi-asserted-by":"crossref","first-page":"531","DOI":"10.1016\/j.bmc.2013.10.045","volume":"22","author":"Del Prete","year":"2014","journal-title":"Bioorg Med Chem"},{"key":"10.1016\/j.bmc.2016.11.021_b0270","doi-asserted-by":"crossref","first-page":"4421","DOI":"10.1021\/cr200176r","volume":"112","author":"Alterio","year":"2012","journal-title":"Chem Rev"},{"key":"10.1016\/j.bmc.2016.11.021_b0275","doi-asserted-by":"crossref","first-page":"680","DOI":"10.1038\/227680a0","volume":"227","author":"Laemmli","year":"1970","journal-title":"Nature"},{"key":"10.1016\/j.bmc.2016.11.021_b0280","doi-asserted-by":"crossref","first-page":"1792","DOI":"10.1093\/nar\/gkh340","volume":"32","author":"Edgar","year":"2004","journal-title":"Nucleic Acids Res"},{"key":"10.1016\/j.bmc.2016.11.021_b0285","doi-asserted-by":"crossref","first-page":"W557","DOI":"10.1093\/nar\/gki352","volume":"33","author":"Guindon","year":"2005","journal-title":"Nucleic Acids Res"}],"container-title":["Bioorganic &amp; Medicinal Chemistry"],"original-title":[],"language":"en","link":[{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0968089616309634?httpAccept=text\/xml","content-type":"text\/xml","content-version":"vor","intended-application":"text-mining"},{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0968089616309634?httpAccept=text\/plain","content-type":"text\/plain","content-version":"vor","intended-application":"text-mining"}],"deposited":{"date-parts":[[2025,10,19]],"date-time":"2025-10-19T00:46:03Z","timestamp":1760834763000},"score":1,"resource":{"primary":{"URL":"https:\/\/linkinghub.elsevier.com\/retrieve\/pii\/S0968089616309634"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2017,1]]},"references-count":57,"journal-issue":{"issue":"2","published-print":{"date-parts":[[2017,1]]}},"alternative-id":["S0968089616309634"],"URL":"https:\/\/doi.org\/10.1016\/j.bmc.2016.11.021","relation":{},"ISSN":["0968-0896"],"issn-type":[{"value":"0968-0896","type":"print"}],"subject":[],"published":{"date-parts":[[2017,1]]},"assertion":[{"value":"Elsevier","name":"publisher","label":"This article is maintained by"},{"value":"Anion inhibition profiles of the \u03b3-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei responsible of melioidosis and highly drug resistant to common antibiotics","name":"articletitle","label":"Article Title"},{"value":"Bioorganic & Medicinal Chemistry","name":"journaltitle","label":"Journal Title"},{"value":"https:\/\/doi.org\/10.1016\/j.bmc.2016.11.021","name":"articlelink","label":"CrossRef DOI link to publisher maintained version"},{"value":"article","name":"content_type","label":"Content Type"},{"value":"\u00a9 2016 Elsevier Ltd. All rights reserved.","name":"copyright","label":"Copyright"}]}}