{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2026,10,6]],"date-time":"2026-10-06T10:58:35Z","timestamp":1791284315705,"version":"4.1.0"},"reference-count":36,"publisher":"Elsevier BV","issue":"2","license":[{"start":{"date-parts":[[2012,1,1]],"date-time":"2012-01-01T00:00:00Z","timestamp":1325376000000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/tdm\/userlicense\/1.0\/"},{"start":{"date-parts":[[2012,1,1]],"date-time":"2012-01-01T00:00:00Z","timestamp":1325376000000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/legal\/tdmrep-license"}],"content-domain":{"domain":["elsevier.com","sciencedirect.com"],"crossmark-restriction":true},"short-container-title":["Bioorganic &amp; Medicinal Chemistry Letters"],"published-print":{"date-parts":[[2012,1]]},"DOI":"10.1016\/j.bmcl.2011.11.108","type":"journal-article","created":{"date-parts":[[2011,12,13]],"date-time":"2011-12-13T22:56:06Z","timestamp":1323816966000},"page":"1103-1106","update-policy":"https:\/\/doi.org\/10.1016\/elsevier_cm_policy","source":"Crossref","is-referenced-by-count":33,"title":["Synthesis of new praziquantel analogues: Potential candidates for the treatment of schistosomiasis"],"prefix":"10.1016","volume":"22","author":[{"given":"Partha Sarathi","family":"Sadhu","sequence":"first","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Singam Naveen","family":"Kumar","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Malapaka","family":"Chandrasekharam","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Livia","family":"Pica-Mattoccia","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Donato","family":"Cioli","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Vaidya Jayathirtha","family":"Rao","sequence":"additional","affiliation":[],"role":[{"vocabulary":"crossref","role":"author"}]}],"member":"78","reference":[{"key":"10.1016\/j.bmcl.2011.11.108_b0005","doi-asserted-by":"crossref","first-page":"41","DOI":"10.1016\/S0001-706X(00)00122-4","volume":"77","author":"Chitsulo","year":"2000","journal-title":"Acta Trop."},{"key":"10.1016\/j.bmcl.2011.11.108_b0010","doi-asserted-by":"crossref","first-page":"658","DOI":"10.1016\/S0140-6736(04)15603-1","volume":"363","author":"Savioli","year":"2004","journal-title":"Lancet"},{"key":"10.1016\/j.bmcl.2011.11.108_b0015","doi-asserted-by":"crossref","first-page":"99","DOI":"10.1016\/S0014-4894(03)00024-9","volume":"102","author":"He","year":"2002","journal-title":"Exp. Parasitol."},{"key":"10.1016\/j.bmcl.2011.11.108_b0020","doi-asserted-by":"crossref","first-page":"125","DOI":"10.1016\/S0001-706X(03)00029-9","volume":"86","author":"Van der Werf","year":"2003","journal-title":"Acta Trop."},{"key":"10.1016\/j.bmcl.2011.11.108_b0025","doi-asserted-by":"crossref","first-page":"35","DOI":"10.1016\/0163-7258(95)00026-7","volume":"68","author":"Cioli","year":"1995","journal-title":"Pharmacol. Ther."},{"key":"10.1016\/j.bmcl.2011.11.108_b0030","doi-asserted-by":"crossref","first-page":"509","DOI":"10.1016\/j.pt.2003.09.005","volume":"19","author":"Fenwick","year":"2003","journal-title":"Trends. Parasitol."},{"key":"10.1016\/j.bmcl.2011.11.108_b0035","doi-asserted-by":"crossref","first-page":"778","DOI":"10.4269\/ajtmh.2004.71.778","volume":"71","author":"Tchuent\u00e9","year":"2004","journal-title":"Am. J. Trop. Hyg."},{"key":"10.1016\/j.bmcl.2011.11.108_b0040","doi-asserted-by":"crossref","first-page":"659","DOI":"10.1097\/00001432-200012000-00014","volume":"13","author":"Cioli","year":"2000","journal-title":"Curr. Opin. Infect. Dis."},{"key":"10.1016\/j.bmcl.2011.11.108_b0045","doi-asserted-by":"crossref","first-page":"458","DOI":"10.5694\/j.1326-5377.1996.tb138598.x","volume":"165","author":"Murray-Smith","year":"1996","journal-title":"Med. J. Aust."},{"key":"10.1016\/j.bmcl.2011.11.108_b0050","doi-asserted-by":"crossref","first-page":"s121","DOI":"10.1016\/j.actatropica.2010.08.020","volume":"120s","author":"Utzinger","year":"2011","journal-title":"Acta. Trop."},{"key":"10.1016\/j.bmcl.2011.11.108_b0055","doi-asserted-by":"crossref","first-page":"e478","DOI":"10.1371\/journal.pntd.0000478","volume":"3","author":"Abdulla","year":"2009","journal-title":"PLoS Negl. Trop. Dis."},{"key":"10.1016\/j.bmcl.2011.11.108_b0060","doi-asserted-by":"crossref","first-page":"e14","DOI":"10.1371\/journal.pmed.0040014","volume":"4","author":"Abdulla","year":"2007","journal-title":"PLoS Med."},{"key":"10.1016\/j.bmcl.2011.11.108_b0065","doi-asserted-by":"crossref","first-page":"e504","DOI":"10.1371\/journal.pntd.0000504","volume":"3","author":"Melman","year":"2009","journal-title":"PLoS Negl. Trop. Dis."},{"key":"10.1016\/j.bmcl.2011.11.108_b0070","doi-asserted-by":"crossref","first-page":"1036","DOI":"10.1007\/BF01945954","volume":"33","author":"Seubert","year":"1977","journal-title":"Experientia"},{"key":"10.1016\/j.bmcl.2011.11.108_b0075","doi-asserted-by":"crossref","first-page":"1731","DOI":"10.3987\/R-1983-09-1731","volume":"20","author":"Frehel","year":"1983","journal-title":"Heterocycles"},{"key":"10.1016\/j.bmcl.2011.11.108_b0080","doi-asserted-by":"crossref","first-page":"5269","DOI":"10.1021\/jo00200a057","volume":"49","author":"Berkowitz","year":"1984","journal-title":"J. Org. Chem."},{"key":"10.1016\/j.bmcl.2011.11.108_b0085","doi-asserted-by":"crossref","first-page":"189","DOI":"10.1002\/jhet.5570230139","volume":"23","author":"Yuste","year":"1986","journal-title":"Heterocyl. Chem."},{"key":"10.1016\/j.bmcl.2011.11.108_b0090","doi-asserted-by":"crossref","first-page":"7395","DOI":"10.1016\/S0040-4020(98)00401-3","volume":"54","author":"Kim","year":"1998","journal-title":"Tetrahedron"},{"key":"10.1016\/j.bmcl.2011.11.108_b0095","doi-asserted-by":"crossref","first-page":"3985","DOI":"10.1021\/jo010990m","volume":"67","author":"Todd","year":"2002","journal-title":"J. Org. Chem."},{"key":"10.1016\/j.bmcl.2011.11.108_b0100","unstructured":"Seubert, J.; Thomas, H.; Andrews, P. German Patent 2, 362, 539, 1975."},{"key":"10.1016\/j.bmcl.2011.11.108_b0105","doi-asserted-by":"crossref","first-page":"186","DOI":"10.3184\/0308234041640564","author":"Ma","year":"2004","journal-title":"Chem. Res."},{"key":"10.1016\/j.bmcl.2011.11.108_b0110","first-page":"17","volume":"2006","author":"Roszkowski","year":"1415","journal-title":"Tetrahedron: Asymmetry"},{"key":"10.1016\/j.bmcl.2011.11.108_b0115","doi-asserted-by":"crossref","first-page":"1287","DOI":"10.1016\/j.tetlet.2005.12.073","volume":"47","author":"El-Fayyoumy","year":"2006","journal-title":"Tetrahedron Lett."},{"key":"10.1016\/j.bmcl.2011.11.108_b0120","doi-asserted-by":"crossref","first-page":"147","DOI":"10.1002\/med.2610030204","volume":"3","author":"Andrews","year":"1983","journal-title":"Med. Res. Rev."},{"key":"10.1016\/j.bmcl.2011.11.108_b0125","doi-asserted-by":"crossref","first-page":"4154","DOI":"10.1016\/j.bmcl.2007.05.063","volume":"17","author":"Ronketti","year":"2007","journal-title":"Biorg.Med. Chem. Lett."},{"key":"10.1016\/j.bmcl.2011.11.108_b0130","doi-asserted-by":"crossref","first-page":"2481","DOI":"10.1016\/j.bmcl.2010.03.001","volume":"20","author":"Dong","year":"2010","journal-title":"Biorg. Med. Chem. Lett."},{"key":"10.1016\/j.bmcl.2011.11.108_b0135_1","doi-asserted-by":"crossref","first-page":"4600","DOI":"10.1016\/j.bmc.2006.02.020","volume":"14","author":"Narender","year":"2006","journal-title":"Bioorg. Med. Chem."},{"key":"10.1016\/j.bmcl.2011.11.108_b0145","doi-asserted-by":"crossref","first-page":"5378","DOI":"10.1016\/j.bmcl.2005.09.008","volume":"15","author":"Narender","year":"2005","journal-title":"Bioorg. Med. Chem. Lett."},{"key":"10.1016\/j.bmcl.2011.11.108_b0150","doi-asserted-by":"crossref","first-page":"3038","DOI":"10.1039\/b306159k","author":"Elliott","year":"2003","journal-title":"Org. Bio. Chem."},{"key":"10.1016\/j.bmcl.2011.11.108_b0155","doi-asserted-by":"crossref","first-page":"3911","DOI":"10.1002\/ejoc.200700261","author":"Werner","year":"2007","journal-title":"Euro. J. Org. Chem."},{"key":"10.1016\/j.bmcl.2011.11.108_b0160","doi-asserted-by":"crossref","first-page":"85","DOI":"10.1039\/j39690000085","author":"Whittaker","year":"1969","journal-title":"Chem. Soc. C"},{"key":"10.1016\/j.bmcl.2011.11.108_b0165","first-page":"1107","volume":"8","author":"Sergovskaya","year":"1991","journal-title":"Khim. Geterotsikl. Soedin."},{"key":"10.1016\/j.bmcl.2011.11.108_b0170","doi-asserted-by":"crossref","first-page":"6895","DOI":"10.1021\/jo900986z","volume":"74","author":"Liu","year":"2009","journal-title":"J. Org. Chem."},{"key":"10.1016\/j.bmcl.2011.11.108_b0175","doi-asserted-by":"crossref","first-page":"e357","DOI":"10.1371\/journal.pntd.0000357","volume":"3","author":"Meyer","year":"2009","journal-title":"PLoS Negl. Trop. Dis."},{"key":"10.1016\/j.bmcl.2011.11.108_b0180","doi-asserted-by":"crossref","first-page":"527","DOI":"10.1016\/j.ijpara.2003.12.003","volume":"34","author":"Pica-Mattoccia","year":"2004","journal-title":"Int. J. Parasitol."},{"key":"10.1016\/j.bmcl.2011.11.108_b0185","unstructured":"For compounds 33\u201337 presence of rotamers were observed in 13C NMR spectrum. So the data for the major isomer only is being reported."}],"container-title":["Bioorganic &amp; Medicinal Chemistry Letters"],"original-title":[],"language":"en","link":[{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0960894X11016520?httpAccept=text\/xml","content-type":"text\/xml","content-version":"vor","intended-application":"text-mining"},{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0960894X11016520?httpAccept=text\/plain","content-type":"text\/plain","content-version":"vor","intended-application":"text-mining"}],"deposited":{"date-parts":[[2025,10,18]],"date-time":"2025-10-18T06:28:43Z","timestamp":1760768923000},"score":1,"resource":{"primary":{"URL":"https:\/\/linkinghub.elsevier.com\/retrieve\/pii\/S0960894X11016520"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2012,1]]},"references-count":36,"journal-issue":{"issue":"2","published-print":{"date-parts":[[2012,1]]}},"alternative-id":["S0960894X11016520"],"URL":"https:\/\/doi.org\/10.1016\/j.bmcl.2011.11.108","relation":{},"ISSN":["0960-894X"],"issn-type":[{"value":"0960-894X","type":"print"}],"subject":[],"published":{"date-parts":[[2012,1]]},"assertion":[{"value":"Elsevier","name":"publisher","label":"This article is maintained by"},{"value":"Synthesis of new praziquantel analogues: Potential candidates for the treatment of schistosomiasis","name":"articletitle","label":"Article Title"},{"value":"Bioorganic & Medicinal Chemistry Letters","name":"journaltitle","label":"Journal Title"},{"value":"https:\/\/doi.org\/10.1016\/j.bmcl.2011.11.108","name":"articlelink","label":"CrossRef DOI link to publisher maintained version"},{"value":"article","name":"content_type","label":"Content Type"},{"value":"Copyright \u00a9 2011 Elsevier Ltd. All rights reserved.","name":"copyright","label":"Copyright"}]}}