{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2026,4,30]],"date-time":"2026-04-30T16:34:26Z","timestamp":1777566866639,"version":"3.51.4"},"reference-count":14,"publisher":"Elsevier BV","license":[{"start":{"date-parts":[[2023,2,1]],"date-time":"2023-02-01T00:00:00Z","timestamp":1675209600000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/tdm\/userlicense\/1.0\/"},{"start":{"date-parts":[[2023,2,1]],"date-time":"2023-02-01T00:00:00Z","timestamp":1675209600000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/legal\/tdmrep-license"},{"start":{"date-parts":[[2023,2,1]],"date-time":"2023-02-01T00:00:00Z","timestamp":1675209600000},"content-version":"stm-asf","delay-in-days":0,"URL":"https:\/\/doi.org\/10.15223\/policy-017"},{"start":{"date-parts":[[2023,2,1]],"date-time":"2023-02-01T00:00:00Z","timestamp":1675209600000},"content-version":"stm-asf","delay-in-days":0,"URL":"https:\/\/doi.org\/10.15223\/policy-037"},{"start":{"date-parts":[[2023,2,1]],"date-time":"2023-02-01T00:00:00Z","timestamp":1675209600000},"content-version":"stm-asf","delay-in-days":0,"URL":"https:\/\/doi.org\/10.15223\/policy-012"},{"start":{"date-parts":[[2023,2,1]],"date-time":"2023-02-01T00:00:00Z","timestamp":1675209600000},"content-version":"stm-asf","delay-in-days":0,"URL":"https:\/\/doi.org\/10.15223\/policy-029"},{"start":{"date-parts":[[2023,2,1]],"date-time":"2023-02-01T00:00:00Z","timestamp":1675209600000},"content-version":"stm-asf","delay-in-days":0,"URL":"https:\/\/doi.org\/10.15223\/policy-004"}],"content-domain":{"domain":["elsevier.com","sciencedirect.com"],"crossmark-restriction":true},"short-container-title":["Bioorganic &amp; Medicinal Chemistry Letters"],"published-print":{"date-parts":[[2023,2]]},"DOI":"10.1016\/j.bmcl.2023.129164","type":"journal-article","created":{"date-parts":[[2023,1,31]],"date-time":"2023-01-31T02:56:02Z","timestamp":1675133762000},"page":"129164","update-policy":"https:\/\/doi.org\/10.1016\/elsevier_cm_policy","source":"Crossref","is-referenced-by-count":8,"special_numbering":"C","title":["Activity of N-phenylbenzamide analogs against the neglected disease pathogen, Schistosoma mansoni"],"prefix":"10.1016","volume":"82","author":[{"ORCID":"https:\/\/orcid.org\/0000-0002-4863-370X","authenticated-orcid":false,"given":"Masebe","family":"Kanyanta","sequence":"first","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Chilufya","family":"Lengwe","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"ORCID":"https:\/\/orcid.org\/0000-0003-4910-4479","authenticated-orcid":false,"given":"Dickson","family":"Mambwe","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"ORCID":"https:\/\/orcid.org\/0000-0001-9742-8801","authenticated-orcid":false,"given":"Karol R.","family":"Francisco","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Lawrence J.","family":"Liu","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Yujie","family":"Uli Sun","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Dilini K.","family":"Amarasinghe","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Conor R.","family":"Caffrey","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]},{"given":"Peter","family":"Mubanga Cheuka","sequence":"additional","affiliation":[],"role":[{"role":"author","vocabulary":"crossref"}]}],"member":"78","reference":[{"key":"10.1016\/j.bmcl.2023.129164_b0005","unstructured":"Schistosomiasis. https:\/\/www.cdc.gov\/dpdx\/schistosomiasis\/index.html (accessed 2022-11-22)."},{"key":"10.1016\/j.bmcl.2023.129164_b0010","unstructured":"Schistosomiasis (Bilharzia). https:\/\/www.who.int\/health-topics\/schistosomiasis (accessed 2022-11-22)."},{"key":"10.1016\/j.bmcl.2023.129164_b0015","unstructured":"WHO factsheet. https:\/\/www.who.int\/news-room\/fact-sheets\/detail\/schistosomiasis (accessed 2022-11-22)."},{"key":"10.1016\/j.bmcl.2023.129164_b0020","first-page":"1","article-title":"Alternatives to praziquantel for the prevention and control of schistosomiasis","volume":"7","author":"Spangenberg","year":"2020","journal-title":"ACS Infect Dis"},{"key":"10.1016\/j.bmcl.2023.129164_b0025","doi-asserted-by":"crossref","first-page":"1595","DOI":"10.2174\/1568026621666210924101805","article-title":"Drug discovery and target identification against schistosomiasis: a reality check on progress and future prospects","volume":"22","author":"Cheuka","year":"2022","journal-title":"Curr Top in Med Chem"},{"key":"10.1016\/j.bmcl.2023.129164_b0030","first-page":"1","article-title":"Early antischistosomal leads identified from in Vitro and in Vivo screening of the medicines for malaria venture pathogen box","volume":"5","author":"Pasche","year":"2018","journal-title":"ACS Infect Dis"},{"key":"10.1016\/j.bmcl.2023.129164_b0035","doi-asserted-by":"crossref","first-page":"1","DOI":"10.1186\/s13071-019-3747-6","article-title":"Multi-center screening of the pathogen box collection for schistosomiasis drug discovery","volume":"12","author":"Maccesi","year":"2019","journal-title":"Parasit Vect"},{"key":"10.1016\/j.bmcl.2023.129164_b0040","first-page":"1","article-title":"Quantitative structure activity relationship in drug design: an overview","volume":"2","author":"Kapoor","year":"2019","journal-title":"SF J Pharm Anal Chem"},{"key":"10.1016\/j.bmcl.2023.129164_b0045","series-title":"Synthesis of ester and amide derivatives of certain NSAIDS","author":"Tegeli","year":"2015"},{"key":"10.1016\/j.bmcl.2023.129164_b0050","doi-asserted-by":"crossref","first-page":"2762","DOI":"10.1016\/j.tet.2018.04.041","article-title":"A method for C2 acylation of 1,3-indandiones","volume":"74","author":"Larsen","year":"2018","journal-title":"Tetrahedron"},{"key":"10.1016\/j.bmcl.2023.129164_b0055","doi-asserted-by":"crossref","first-page":"28","DOI":"10.1016\/j.ejphar.2017.02.051","article-title":"Molecular docking, synthesis and biological screening of mefenamic acid derivatives as anti-inflammatory agents","volume":"801","author":"Savjani","year":"2017","journal-title":"Eur J Pharmacol"},{"key":"10.1016\/j.bmcl.2023.129164_b0060","doi-asserted-by":"crossref","first-page":"1","DOI":"10.1371\/journal.pntd.0004356","article-title":"Structure-bioactivity relationship for benzimidazole thiophene inhibitors of polo-like kinase 1 (PLK1), a potential drug target in Schistosoma mansoni","volume":"10","author":"Long","year":"2016","journal-title":"PLoS Neglect Trop Dis"},{"key":"10.1016\/j.bmcl.2023.129164_b0065","doi-asserted-by":"crossref","first-page":"258","DOI":"10.1021\/acsmedchemlett.9b00455","article-title":"Structure-bioactivity relationships of lapatinib derived analogs against Schistosoma mansoni","volume":"11","author":"Buskes","year":"2020","journal-title":"ACS Med Chem Lett"},{"key":"10.1016\/j.bmcl.2023.129164_b0070","doi-asserted-by":"crossref","first-page":"1935","DOI":"10.1128\/AAC.04463-14","article-title":"Activities of N, N\u2032-Diarylurea MMV665852 analogs against Schistosoma mansoni","volume":"59","author":"Cowan","year":"2015","journal-title":"Antimicrob Agents Chemother"}],"container-title":["Bioorganic &amp; Medicinal Chemistry Letters"],"original-title":[],"language":"en","link":[{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0960894X23000422?httpAccept=text\/xml","content-type":"text\/xml","content-version":"vor","intended-application":"text-mining"},{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0960894X23000422?httpAccept=text\/plain","content-type":"text\/plain","content-version":"vor","intended-application":"text-mining"}],"deposited":{"date-parts":[[2025,10,18]],"date-time":"2025-10-18T07:46:24Z","timestamp":1760773584000},"score":1,"resource":{"primary":{"URL":"https:\/\/linkinghub.elsevier.com\/retrieve\/pii\/S0960894X23000422"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2023,2]]},"references-count":14,"alternative-id":["S0960894X23000422"],"URL":"https:\/\/doi.org\/10.1016\/j.bmcl.2023.129164","relation":{},"ISSN":["0960-894X"],"issn-type":[{"value":"0960-894X","type":"print"}],"subject":[],"published":{"date-parts":[[2023,2]]},"assertion":[{"value":"Elsevier","name":"publisher","label":"This article is maintained by"},{"value":"Activity of N-phenylbenzamide analogs against the neglected disease pathogen, Schistosoma mansoni","name":"articletitle","label":"Article Title"},{"value":"Bioorganic & Medicinal Chemistry Letters","name":"journaltitle","label":"Journal Title"},{"value":"https:\/\/doi.org\/10.1016\/j.bmcl.2023.129164","name":"articlelink","label":"CrossRef DOI link to publisher maintained version"},{"value":"article","name":"content_type","label":"Content Type"},{"value":"\u00a9 2023 Elsevier Ltd. All rights reserved.","name":"copyright","label":"Copyright"}],"article-number":"129164"}}