{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2026,4,9]],"date-time":"2026-04-09T16:26:28Z","timestamp":1775751988881,"version":"3.50.1"},"reference-count":38,"publisher":"Elsevier BV","issue":"23","license":[{"start":{"date-parts":[[2013,12,1]],"date-time":"2013-12-01T00:00:00Z","timestamp":1385856000000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/tdm\/userlicense\/1.0\/"},{"start":{"date-parts":[[2013,12,1]],"date-time":"2013-12-01T00:00:00Z","timestamp":1385856000000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/legal\/tdmrep-license"}],"content-domain":{"domain":["elsevier.com","sciencedirect.com"],"crossmark-restriction":true},"short-container-title":["Bioorganic &amp; Medicinal Chemistry Letters"],"published-print":{"date-parts":[[2013,12]]},"DOI":"10.1016\/j.bmcl.2013.09.047","type":"journal-article","created":{"date-parts":[[2013,9,25]],"date-time":"2013-09-25T06:50:37Z","timestamp":1380091837000},"page":"6436-6441","update-policy":"https:\/\/doi.org\/10.1016\/elsevier_cm_policy","source":"Crossref","is-referenced-by-count":54,"title":["Synthesis and anti-parasitic activity of a novel quinolinone\u2013chalcone series"],"prefix":"10.1016","volume":"23","author":[{"given":"Marina","family":"Roussaki","sequence":"first","affiliation":[]},{"given":"Belinda","family":"Hall","sequence":"additional","affiliation":[]},{"given":"Sofia Costa","family":"Lima","sequence":"additional","affiliation":[]},{"given":"Anabela Cordeiro","family":"da Silva","sequence":"additional","affiliation":[]},{"given":"Shane","family":"Wilkinson","sequence":"additional","affiliation":[]},{"given":"Anastasia","family":"Detsi","sequence":"additional","affiliation":[]}],"member":"78","reference":[{"key":"10.1016\/j.bmcl.2013.09.047_b0005","unstructured":"Crompton, D. W.T, In Sustaining the drive to overcome the global impact of neglected tropical diseases, Second WHO report on neglected tropical diseases, 2013, WHO reference number: WHO\/HTM\/NTD\/2013.1."},{"key":"10.1016\/j.bmcl.2013.09.047_b0010","doi-asserted-by":"crossref","first-page":"1301","DOI":"10.1172\/JCI33945","volume":"118","author":"Stuart","year":"2008","journal-title":"J. Clin. Invest."},{"key":"10.1016\/j.bmcl.2013.09.047_b0015","doi-asserted-by":"crossref","first-page":"2893","DOI":"10.1128\/AAC.00332-10","volume":"54","author":"Sokolova","year":"2010","journal-title":"Antimicrob. Agents Chemother."},{"key":"10.1016\/j.bmcl.2013.09.047_b0020","doi-asserted-by":"crossref","first-page":"411","DOI":"10.1007\/s00415-006-0093-3","volume":"253","author":"Kennedy","year":"2006","journal-title":"J. Neurol."},{"key":"10.1016\/j.bmcl.2013.09.047_b0025","doi-asserted-by":"crossref","first-page":"55","DOI":"10.1371\/journal.pmed.0050055","volume":"5","author":"Simarro","year":"2008","journal-title":"PLoS Med."},{"key":"10.1016\/j.bmcl.2013.09.047_b0030","doi-asserted-by":"crossref","first-page":"148","DOI":"10.1016\/S0140-6736(09)60829-1","volume":"375","author":"Brun","year":"2010","journal-title":"Lancet"},{"key":"10.1016\/j.bmcl.2013.09.047_b0035","first-page":"12","volume":"3","author":"Steverding","year":"2008","journal-title":"Parasite Vector"},{"key":"10.1016\/j.bmcl.2013.09.047_b0040","doi-asserted-by":"crossref","first-page":"502","DOI":"10.1016\/j.pt.2003.09.008","volume":"19","author":"Croft","year":"2003","journal-title":"Trends Parasitol."},{"key":"10.1016\/j.bmcl.2013.09.047_b0045","doi-asserted-by":"crossref","first-page":"1","DOI":"10.2174\/157488410790410579","volume":"5","author":"Batovska","year":"2010","journal-title":"Curr. Clin. Pharmacol."},{"key":"10.1016\/j.bmcl.2013.09.047_b0050","doi-asserted-by":"crossref","first-page":"186","DOI":"10.2174\/092986713804806630","volume":"20","author":"Roman","year":"2013","journal-title":"Curr. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0055","doi-asserted-by":"crossref","first-page":"435","DOI":"10.1016\/j.ejmech.2013.01.018","volume":"62","author":"Shenvi","year":"2013","journal-title":"Eur. J. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0060","doi-asserted-by":"crossref","first-page":"8073","DOI":"10.1016\/j.bmc.2009.10.002","volume":"17","author":"Detsi","year":"2009","journal-title":"Bioorg. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0065","doi-asserted-by":"crossref","first-page":"259","DOI":"10.1016\/j.phrs.2008.02.005","volume":"57","author":"Mojzis","year":"2008","journal-title":"Pharmacol. Res."},{"key":"10.1016\/j.bmcl.2013.09.047_b0070","doi-asserted-by":"crossref","first-page":"125","DOI":"10.1016\/j.ejmech.2006.09.019","volume":"42","author":"Nowakowska","year":"2007","journal-title":"Eur. J. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0075","doi-asserted-by":"crossref","first-page":"51","DOI":"10.1016\/j.ejmech.2013.04.056","volume":"65","author":"Bano","year":"2013","journal-title":"Eur. J. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0080","doi-asserted-by":"crossref","first-page":"S55","DOI":"10.1007\/s00436-002-0768-3","volume":"90","author":"Kayser","year":"2003","journal-title":"Parasitol. Res."},{"key":"10.1016\/j.bmcl.2013.09.047_b0085","doi-asserted-by":"crossref","first-page":"2023","DOI":"10.1128\/AAC.45.7.2023-2029.2001","volume":"45","author":"Chen","year":"2001","journal-title":"Antimicrob. Agents Chemother."},{"key":"10.1016\/j.bmcl.2013.09.047_b0090","doi-asserted-by":"crossref","first-page":"396","DOI":"10.1016\/j.ejmech.2013.03.065","volume":"64","author":"Ryczak","year":"2013","journal-title":"Eur. J. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0095","doi-asserted-by":"crossref","first-page":"291","DOI":"10.1016\/j.bmcl.2012.10.101","volume":"23","author":"Tyagi","year":"2013","journal-title":"Bioorg. Med. Chem. Lett."},{"key":"10.1016\/j.bmcl.2013.09.047_b0100","doi-asserted-by":"crossref","first-page":"3553","DOI":"10.1021\/jm2012408","volume":"55","author":"Qiao","year":"2012","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0105","doi-asserted-by":"crossref","first-page":"1397","DOI":"10.1021\/np058018g","volume":"68","author":"He","year":"2005","journal-title":"J. Nat. Prod."},{"key":"10.1016\/j.bmcl.2013.09.047_b0110","doi-asserted-by":"crossref","first-page":"2421","DOI":"10.1016\/j.tet.2012.01.007","volume":"68","author":"Nakashima","year":"2012","journal-title":"Tetrahedron"},{"key":"10.1016\/j.bmcl.2013.09.047_b0115","doi-asserted-by":"crossref","first-page":"1458","DOI":"10.1248\/cpb.c12-00487","volume":"60","author":"Gao","year":"2012","journal-title":"Chem. Pharm. Bull."},{"key":"10.1016\/j.bmcl.2013.09.047_b0120","doi-asserted-by":"crossref","first-page":"2325","DOI":"10.1016\/j.tetlet.2013.02.081","volume":"54","author":"Angeleska","year":"2013","journal-title":"Tetrahedron Lett."},{"key":"10.1016\/j.bmcl.2013.09.047_b0125","doi-asserted-by":"crossref","first-page":"2450","DOI":"10.1021\/jm061173n","volume":"50","author":"Detsi","year":"2007","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0130","doi-asserted-by":"crossref","first-page":"2075","DOI":"10.1021\/jm031044w","volume":"47","author":"Jonsson","year":"2004","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0135","doi-asserted-by":"crossref","first-page":"4497","DOI":"10.1021\/jm400211f","volume":"56","author":"Larsson","year":"2013","journal-title":"J. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0140","doi-asserted-by":"crossref","first-page":"317","DOI":"10.1016\/0031-9422(95)00265-9","volume":"40","author":"Lavaud","year":"1995","journal-title":"Phytochemistry"},{"key":"10.1016\/j.bmcl.2013.09.047_b0145","doi-asserted-by":"crossref","first-page":"44","DOI":"10.1016\/j.ejmech.2012.03.003","volume":"52","author":"Audisio","year":"2012","journal-title":"Eur. J. Med. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0150","doi-asserted-by":"crossref","first-page":"2909","DOI":"10.1039\/p19960002909","author":"Detsi","year":"1996","journal-title":"J. Chem. Soc., Perkin Trans. 1"},{"key":"10.1016\/j.bmcl.2013.09.047_b0155","doi-asserted-by":"crossref","first-page":"1257","DOI":"10.1023\/A:1013229213478","volume":"71","author":"Kalechits","year":"2001","journal-title":"Russ. J. Gen. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0160","first-page":"171","volume":"16","author":"Sarveswari","year":"2006","journal-title":"Ind. J. Heterocycl. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0165","first-page":"4215","volume":"23","author":"Bhupathi","year":"2011","journal-title":"Asian J. Chem."},{"key":"10.1016\/j.bmcl.2013.09.047_b0170","unstructured":"Boyle, R. G.; Imogai, H. J.; Cherry, M.; Humphries, A. J., Navarro, E. F.; Owen, D. R.; Dales, N. A.; Lamarche, M.; Cullis, C., Gould, A. E. WO 2005\/028474 A2."},{"key":"10.1016\/j.bmcl.2013.09.047_b0175","doi-asserted-by":"crossref","first-page":"407","DOI":"10.1111\/j.1747-0285.2010.01020.x","volume":"76","author":"Sivakumar","year":"2010","journal-title":"Chem. Biol. Drug Des."},{"key":"10.1016\/j.bmcl.2013.09.047_b0180","doi-asserted-by":"crossref","first-page":"915","DOI":"10.1101\/gr.115089.110","volume":"21","author":"Alsford","year":"2011","journal-title":"Genome Res."},{"key":"10.1016\/j.bmcl.2013.09.047_b0185","doi-asserted-by":"crossref","first-page":"1636","DOI":"10.1093\/carcin\/bgt087","volume":"34","author":"Wu","year":"2013","journal-title":"Carcinogenesis"},{"key":"10.1016\/j.bmcl.2013.09.047_b0190","doi-asserted-by":"crossref","first-page":"323","DOI":"10.1042\/BJ20061281","volume":"403","author":"Piacenza","year":"2007","journal-title":"Biochem. J."}],"container-title":["Bioorganic &amp; Medicinal Chemistry Letters"],"original-title":[],"language":"en","link":[{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0960894X13011219?httpAccept=text\/xml","content-type":"text\/xml","content-version":"vor","intended-application":"text-mining"},{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S0960894X13011219?httpAccept=text\/plain","content-type":"text\/plain","content-version":"vor","intended-application":"text-mining"}],"deposited":{"date-parts":[[2025,10,18]],"date-time":"2025-10-18T06:48:08Z","timestamp":1760770088000},"score":1,"resource":{"primary":{"URL":"https:\/\/linkinghub.elsevier.com\/retrieve\/pii\/S0960894X13011219"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2013,12]]},"references-count":38,"journal-issue":{"issue":"23","published-print":{"date-parts":[[2013,12]]}},"alternative-id":["S0960894X13011219"],"URL":"https:\/\/doi.org\/10.1016\/j.bmcl.2013.09.047","relation":{},"ISSN":["0960-894X"],"issn-type":[{"value":"0960-894X","type":"print"}],"subject":[],"published":{"date-parts":[[2013,12]]},"assertion":[{"value":"Elsevier","name":"publisher","label":"This article is maintained by"},{"value":"Synthesis and anti-parasitic activity of a novel quinolinone\u2013chalcone series","name":"articletitle","label":"Article Title"},{"value":"Bioorganic & Medicinal Chemistry Letters","name":"journaltitle","label":"Journal Title"},{"value":"https:\/\/doi.org\/10.1016\/j.bmcl.2013.09.047","name":"articlelink","label":"CrossRef DOI link to publisher maintained version"},{"value":"article","name":"content_type","label":"Content Type"},{"value":"Copyright \u00a9 2013 Elsevier Ltd. Published by Elsevier Ltd. All rights reserved.","name":"copyright","label":"Copyright"}]}}