{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2023,6,12]],"date-time":"2023-06-12T22:27:57Z","timestamp":1686608877214},"reference-count":56,"publisher":"Elsevier BV","issue":"1-3","license":[{"start":{"date-parts":[[2001,6,1]],"date-time":"2001-06-01T00:00:00Z","timestamp":991353600000},"content-version":"tdm","delay-in-days":0,"URL":"https:\/\/www.elsevier.com\/tdm\/userlicense\/1.0\/"}],"content-domain":{"domain":[],"crossmark-restriction":false},"short-container-title":["European Journal of Pharmacology"],"published-print":{"date-parts":[[2001,6]]},"DOI":"10.1016\/s0014-2999(01)01055-x","type":"journal-article","created":{"date-parts":[[2002,7,25]],"date-time":"2002-07-25T17:40:30Z","timestamp":1027618830000},"page":"31-37","source":"Crossref","is-referenced-by-count":6,"title":["Effect of P-glycoprotein modulators on the human extraneuronal monoamine transporter"],"prefix":"10.1016","volume":"422","author":[{"given":"F\u00e1tima","family":"Martel","sequence":"first","affiliation":[]},{"given":"Elisa","family":"Keating","sequence":"additional","affiliation":[]},{"given":"Isabel","family":"Azevedo","sequence":"additional","affiliation":[]}],"member":"78","reference":[{"key":"10.1016\/S0014-2999(01)01055-X_BIB1","first-page":"E604","article-title":"Extremity amino acid metabolism during starvation and intravenous feeding in humans","volume":"251","author":"Albert","year":"1986","journal-title":"Am. J. Physiol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB2","doi-asserted-by":"crossref","first-page":"361","DOI":"10.1146\/annurev.pharmtox.39.1.361","article-title":"Biochemical, cellular, and pharmacological aspects of the multidrug transporter","volume":"39","author":"Ambudkar","year":"1999","journal-title":"Annu. Rev. Pharmacol. Toxicol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB3","doi-asserted-by":"crossref","first-page":"161","DOI":"10.1146\/annurev.pa.36.040196.001113","article-title":"P-glycoproteins and multidrug resistance","volume":"36","author":"Bellamy","year":"1996","journal-title":"Annu. Rev. Pharmacol. Toxicol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB4","doi-asserted-by":"crossref","first-page":"659","DOI":"10.1016\/0024-3205(78)90064-4","article-title":"The tyramines: functionally significant biogenic amines or metabolic accidents?","volume":"23","author":"Boulton","year":"1978","journal-title":"Life Sci."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB5","first-page":"179","article-title":"Trace amines in the central nervous system","volume":"26","author":"Boulton","year":"1979","journal-title":"Int. Rev. Biochem."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB6","first-page":"413","article-title":"The tyramines: are they involved in the psychosis?","volume":"14","author":"Boulton","year":"1979","journal-title":"Biol. Psychiatr."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB7","doi-asserted-by":"crossref","first-page":"248","DOI":"10.1016\/0003-2697(76)90527-3","article-title":"A rapid method for the quantitation of microgram quantities of protein utilizing the principle of protein-dye binding","volume":"72","author":"Bradford","year":"1976","journal-title":"Anal. Biochem."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB8","doi-asserted-by":"crossref","first-page":"218","DOI":"10.1038\/sj.bjp.0702065","article-title":"Catecholamine transport by the organic cation transporter type 1 (OCT1)","volume":"125","author":"Breidert","year":"1998","journal-title":"Br. J. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB9","doi-asserted-by":"crossref","first-page":"32599","DOI":"10.1074\/jbc.271.51.32599","article-title":"Electrogenic properties and substrate specificity of the polyspecific rat cation transporter rOCT1","volume":"271","author":"Busch","year":"1996","journal-title":"J. Biol. Chem."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB10","doi-asserted-by":"crossref","first-page":"1389","DOI":"10.1111\/j.1476-5381.1996.tb15550.x","article-title":"Transport and epithelial secretion of the cardiac glycoside, digoxin, by human intestinal epithelial (Caco-2) cells","volume":"118","author":"Cavet","year":"1996","journal-title":"Br. J. Pharmacol."},{"issue":"Suppl. 6","key":"10.1016\/S0014-2999(01)01055-X_BIB11","doi-asserted-by":"crossref","first-page":"53","DOI":"10.1023\/A:1008332318884","article-title":"Modulation of multidrug resistance (MDR) in hematological malignancies","volume":"10","author":"Covelli","year":"1999","journal-title":"Ann. Oncol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB12","doi-asserted-by":"crossref","first-page":"287","DOI":"10.1007\/BF00171059","article-title":"Disprocynium24, a novel inhibitor of the extraneuronal monoamine transporter, has potent effects on the inactivation of circulating noradrenaline and adrenaline in the conscious rat","volume":"354","author":"Eisenhofer","year":"1996","journal-title":"Naunyn-Schmiedeberg's Arch. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB13","doi-asserted-by":"crossref","first-page":"295","DOI":"10.1021\/js970294v","article-title":"Role of P-glycoprotein as a secretory mechanism in quinidine absorption from rat small intestine","volume":"87","author":"Emi","year":"1998","journal-title":"J. Pharm. Sci."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB14","doi-asserted-by":"crossref","first-page":"275","DOI":"10.1007\/BF00171058","article-title":"The role of extraneuronal amine transport systems for the removal of extracellular catecholamines in the rabbit","volume":"354","author":"Friedgen","year":"1996","journal-title":"Naunyn-Schmiedeberg's Arch. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB15","doi-asserted-by":"crossref","first-page":"871","DOI":"10.1089\/dna.1997.16.871","article-title":"Cloning and characterization of two human polyspecific organic cation transporters","volume":"16","author":"Gorboulev","year":"1997","journal-title":"DNA Cell Biol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB16","doi-asserted-by":"crossref","first-page":"59","DOI":"10.1099\/0022-1317-36-1-59","article-title":"Characteristics of a human cell line transformed by DNA from human adenovirus type 5","volume":"36","author":"Graham","year":"1977","journal-title":"J. Gen. Virol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB17","doi-asserted-by":"crossref","first-page":"1556","DOI":"10.1002\/hep.510290530","article-title":"Cloning and functional expression of a mouse liver organic cation transporter","volume":"29","author":"Green","year":"1999","journal-title":"Hepatology"},{"key":"10.1016\/S0014-2999(01)01055-X_BIB18","doi-asserted-by":"crossref","first-page":"30915","DOI":"10.1074\/jbc.273.47.30915","article-title":"Transport of monoamine transmitters by the organic cation transporter type 2, OCT2","volume":"273","author":"Gr\u00fcndemann","year":"1998","journal-title":"J. Biol. Chem."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB19","doi-asserted-by":"crossref","first-page":"349","DOI":"10.1038\/1557","article-title":"Molecular identification of the corticosterone-sensitive extraneuronal monoamine transporter","volume":"1","author":"Gr\u00fcndemann","year":"1998","journal-title":"Nat. Neurosci."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB20","doi-asserted-by":"crossref","first-page":"1","DOI":"10.1124\/mol.56.1.1","article-title":"Selective substrates for non-neuronal monoamine transporters","volume":"56","author":"Gr\u00fcndemann","year":"1999","journal-title":"Mol. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB21","doi-asserted-by":"crossref","first-page":"83","DOI":"10.1016\/0304-3940(89)90445-X","article-title":"The biodisposition of MPP+ in mouse brain","volume":"101","author":"Irwin","year":"1989","journal-title":"Neurosci. Lett."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB22","first-page":"18","article-title":"The uptake of catechol amines at high perfusion concentrations in the isolated rat heart: a novel catechol amine uptake process","volume":"25","author":"Iversen","year":"1965","journal-title":"Br. J. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB23","doi-asserted-by":"crossref","first-page":"15971","DOI":"10.1074\/jbc.273.26.15971","article-title":"Cloning and functional characterization of a potential-sensitive, polyspecific organic cation transporter (OCT3) most abundantly expressed in placenta","volume":"273","author":"Kekuda","year":"1998","journal-title":"J. Biol. Chem."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB24","series-title":"Mammalian Amino Acid Transport: Mechanisms and Control","first-page":"195","article-title":"Muscle amino acid metabolism and transport","author":"Mackenzie","year":"1992"},{"key":"10.1016\/S0014-2999(01)01055-X_BIB25","doi-asserted-by":"crossref","first-page":"1519","DOI":"10.1111\/j.1476-5381.1996.tb16067.x","article-title":"Inward transport of 3H-1-methyl-4-phenylpyridinium (MPP+) in isolated rat hepatocytes: putative involvement of a P-glycoprotein transporter","volume":"119","author":"Martel","year":"1996","journal-title":"Br. J. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB26","doi-asserted-by":"crossref","first-page":"57","DOI":"10.1046\/j.1365-2680.1998.1810057.x","article-title":"Uptake of 3H-adrenaline by freshly isolated rat hepatocytes: putative involvement of P-glycoprotein","volume":"18","author":"Martel","year":"1998","journal-title":"J. Auton. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB27","doi-asserted-by":"crossref","first-page":"131","DOI":"10.1006\/phrs.1997.0283","article-title":"Postnatal development of organic cation transport in the rat liver","volume":"37","author":"Martel","year":"1998","journal-title":"Pharmacol. Res."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB28","doi-asserted-by":"crossref","first-page":"211","DOI":"10.1016\/S0014-2999(99)00501-4","article-title":"Characterization of the efflux of the organic cation MPP+ in cultured rat hepatocytes","volume":"379","author":"Martel","year":"1999","journal-title":"Eur. J. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB29","doi-asserted-by":"crossref","first-page":"505","DOI":"10.1007\/s002100000223","article-title":"Characterization of the transport of the organic cation [3H]-MPP+ in human intestinal epithelial (Caco-2) cells","volume":"361","author":"Martel","year":"2000","journal-title":"Naunyn-Schmiedeberg's Arch. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB30","doi-asserted-by":"crossref","first-page":"1","DOI":"10.1007\/s002100000302","article-title":"Transport of [3H]MPP+ in an immortalized rat brain microvessel endothelial cell line (RBE 4)","volume":"363","author":"Martel","year":"2001","journal-title":"Naunyn-Schmiedeberg's Arch. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB31","doi-asserted-by":"crossref","first-page":"40","DOI":"10.1007\/s002100000335","article-title":"Apical uptake of organic cations by human intestinal Caco-2 cells: putative involvement of ASF transporters","volume":"363","author":"Martel","year":"2001","journal-title":"Naunyn-Schmiedeberg's Arch. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB32","series-title":"Graphpad Prism (version 1.0)","author":"Motulsky","year":"1994"},{"key":"10.1016\/S0014-2999(01)01055-X_BIB33","first-page":"778","article-title":"Na(+)-dependent carnitine transport by organic cation transporter (OCTN2): its pharmacological and toxicological relevance","volume":"291","author":"Ohashi","year":"1999","journal-title":"J. Pharmacol. Exp. Ther."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB34","doi-asserted-by":"crossref","first-page":"366","DOI":"10.1139\/o74-055","article-title":"Identification and distribution of p-tyramine in the rat","volume":"52","author":"Philips","year":"1974","journal-title":"Can. J. Biochem."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB35","doi-asserted-by":"crossref","first-page":"195","DOI":"10.1076\/0271-3683(200003)2031-9FT195","article-title":"Expression of the extraneuronal monoamine transporter in RPE and neural retina","volume":"20","author":"Rajan","year":"2000","journal-title":"Curr. Eye Res."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB36","doi-asserted-by":"crossref","first-page":"85","DOI":"10.1016\/S0005-2736(97)00185-5","article-title":"Effects of cardiovascular drugs on ATPase activity of P-glycoprotein in plasma membranes and in purified reconstituted form","volume":"1369","author":"Rebbeor","year":"1998","journal-title":"Biochim. Biophys. Acta"},{"key":"10.1016\/S0014-2999(01)01055-X_BIB37","doi-asserted-by":"crossref","first-page":"536","DOI":"10.1046\/j.1365-2362.1999.00495.x","article-title":"Multidrug resistance in oncology: diagnostic and therapeutic approaches","volume":"29","author":"Robert","year":"1999","journal-title":"Eur. J. Clin. Invest."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB38","doi-asserted-by":"crossref","first-page":"158","DOI":"10.1007\/BF00165297","article-title":"The extraneuronal transport mechanism for noradrenaline (uptake2) avidly transports 1-methyl-4-phenylpyridinium (MPP+)","volume":"346","author":"Russ","year":"1992","journal-title":"Naunyn-Schmiedeberg's Arch. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB39","doi-asserted-by":"crossref","first-page":"1256","DOI":"10.1111\/j.1460-9568.1996.tb01294.x","article-title":"The extraneuronal transporter for monoamine transmitters exists in cells derived from human central nervous system glia","volume":"8","author":"Russ","year":"1996","journal-title":"Eur. J. Neurosci."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB40","series-title":"Catecholamines II","first-page":"181","article-title":"\u00df-phenylethylamine, phenylethanolamine, tyramine and octopamine","volume":"vol. 90\/II","author":"Saavedra","year":"1989"},{"key":"10.1016\/S0014-2999(01)01055-X_BIB41","doi-asserted-by":"crossref","first-page":"121","DOI":"10.1016\/0378-4274(89)90168-9","article-title":"Biochemical mechanism of action of the dopaminergic neurotoxin 1-methyl-4-phenyl-1,2,3,6-tetrahydropyridine (MPTP)","volume":"48","author":"Sayre","year":"1989","journal-title":"Toxicol. Lett."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB42","doi-asserted-by":"crossref","first-page":"79","DOI":"10.1016\/S0014-5793(98)00203-8","article-title":"Molecular cloning and characterization of two novel transport proteins from rat kidney","volume":"425","author":"Sch\u00f6mig","year":"1998","journal-title":"FEBS Lett."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB43","doi-asserted-by":"crossref","first-page":"868","DOI":"10.1016\/0026-0495(85)90112-X","article-title":"Normal plasma amino acid values in adults: the influence of some common physiological variables","volume":"34","author":"Scriver","year":"1985","journal-title":"Metabolism"},{"key":"10.1016\/S0014-2999(01)01055-X_BIB44","series-title":"Enzyme Kinetics: Behavior and Analysis of Rapid Equilibrium and Steady-State Enzyme Systems","author":"Segel","year":"1975"},{"issue":"Suppl. 6","key":"10.1016\/S0014-2999(01)01055-X_BIB45","doi-asserted-by":"crossref","first-page":"149","DOI":"10.1023\/A:1008355801988","article-title":"New approaches in cancer treatment","volume":"10","author":"Sikic","year":"1999","journal-title":"Ann. Oncol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB46","doi-asserted-by":"crossref","first-page":"361","DOI":"10.1038\/sj.bjp.0701606","article-title":"Interactions between P-glycoprotein substrates and other cationic drugs at the hepatic excretory level","volume":"123","author":"Smit","year":"1998","journal-title":"Br. J. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB47","doi-asserted-by":"crossref","first-page":"521","DOI":"10.1046\/j.1365-2796.2000.t01-1-00689.x","article-title":"Multidrug resistance in haematological malignancies","volume":"247","author":"Sonneveld","year":"2000","journal-title":"J. Intern. Med."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB48","first-page":"R118","article-title":"The extraneuronal noradrenaline carrier (uptake2) exists in the central nervous system (CNS)","volume":"347","author":"Staudt","year":"1993","journal-title":"Naunyn-Schmiedeberg's Arch. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB49","doi-asserted-by":"crossref","first-page":"328","DOI":"10.1007\/BF00168636","article-title":"Expression of the extraneuronal monoamine transporter (uptake2) in human glioma cells","volume":"353","author":"Streich","year":"1996","journal-title":"Naunyn-Schmiedeberg's Arch. Pharmacol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB50","doi-asserted-by":"crossref","first-page":"465","DOI":"10.1111\/j.1471-4159.1976.tb12269.x","article-title":"A sensitive enzymatic-isotopic method for the analysis of tyramine in brain and other tissues","volume":"27","author":"Tallman","year":"1976","journal-title":"J. Neurochem."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB51","series-title":"Catecholamines I","first-page":"279","article-title":"The extraneuronal uptake and metabolism of catecholamines","volume":"vol. 90\/I","author":"Trendelenburg","year":"1988"},{"key":"10.1016\/S0014-2999(01)01055-X_BIB52","doi-asserted-by":"crossref","first-page":"280","DOI":"10.1007\/BF00374179","article-title":"Bisubstrates: substances that interact with renal contraluminal organic anion and organic cation transport systems. I. Amines, piperidines, piperazines, azepines, pyridine, quinolines, imidazoles, thiazoles, guanidines and hydrazines","volume":"425","author":"Ullrich","year":"1993","journal-title":"Pfluegers Arch. Eur. J. Physiol."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB53","first-page":"768","article-title":"Novel membrane transporter OCTN1 mediates multispecific, bidirectional, and pH-dependent transport of organic cations","volume":"289","author":"Yabuuchi","year":"1999","journal-title":"J. Pharmacol. Exp. Ther."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB54","series-title":"Neuroregulators and Psychiatric Disorders","article-title":"Tyramine and Psychiatric disorders","author":"Youdim","year":"1977"},{"key":"10.1016\/S0014-2999(01)01055-X_BIB55","first-page":"354","article-title":"Functional characterization of an organic cation transporter (hOCT1) in a transiently transfected human cell line (HeLa)","volume":"286","author":"Zhang","year":"1998","journal-title":"J. Pharmacol. Exp. Ther."},{"key":"10.1016\/S0014-2999(01)01055-X_BIB56","doi-asserted-by":"crossref","first-page":"2093","DOI":"10.1096\/fasebj.5.7.2010061","article-title":"Choline, an essential nutrient for humans","volume":"5","author":"Zeisel","year":"1991","journal-title":"FASEB J."}],"container-title":["European Journal of Pharmacology"],"original-title":[],"language":"en","link":[{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S001429990101055X?httpAccept=text\/xml","content-type":"text\/xml","content-version":"vor","intended-application":"text-mining"},{"URL":"https:\/\/api.elsevier.com\/content\/article\/PII:S001429990101055X?httpAccept=text\/plain","content-type":"text\/plain","content-version":"vor","intended-application":"text-mining"}],"deposited":{"date-parts":[[2020,1,14]],"date-time":"2020-01-14T17:17:40Z","timestamp":1579022260000},"score":1,"resource":{"primary":{"URL":"https:\/\/linkinghub.elsevier.com\/retrieve\/pii\/S001429990101055X"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2001,6]]},"references-count":56,"journal-issue":{"issue":"1-3","published-print":{"date-parts":[[2001,6]]}},"alternative-id":["S001429990101055X"],"URL":"https:\/\/doi.org\/10.1016\/s0014-2999(01)01055-x","relation":{},"ISSN":["0014-2999"],"issn-type":[{"value":"0014-2999","type":"print"}],"subject":[],"published":{"date-parts":[[2001,6]]}}}