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Chem."],"abstract":"<jats:p>\n                    We report here the synthesis and antibacterial\/antibiofilm activities of 18 sulfa drug analogues with an\u00a0\n                    <jats:italic>N<\/jats:italic>\n                    -acylsulfonamide moiety obtained efficiently by sulfo-click reactions between readily available thioacid and sulfonyl azide synthons.\n                  <\/jats:p>","DOI":"10.1039\/d3md00229b","type":"journal-article","created":{"date-parts":[[2023,7,4]],"date-time":"2023-07-04T09:02:45Z","timestamp":1688461365000},"page":"1567-1571","update-policy":"https:\/\/doi.org\/10.1039\/rsc_crossmark_policy","source":"Crossref","is-referenced-by-count":11,"title":["<i>N<\/i>\n                    -Acylsulfonamide: a valuable moiety to design new sulfa drug analogues"],"prefix":"10.1039","volume":"14","author":[{"ORCID":"https:\/\/orcid.org\/0000-0002-7498-0334","authenticated-orcid":false,"given":"Romain","family":"Amador","sequence":"first","affiliation":[{"name":"Institut des Biomol\u00e9cules Max Mousseron, Universit\u00e9 de Montpellier, CNRS, ENSCM, 1919 route de Mende, 34095 Montpellier, France"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"ORCID":"https:\/\/orcid.org\/0000-0003-4064-820X","authenticated-orcid":false,"given":"Ali","family":"Tahrioui","sequence":"additional","affiliation":[{"name":"Univ Rouen Normandie, Universit\u00e9 Caen Normandie, Normandie Univ, Communication Bact\u00e9rienne et Strat\u00e9gies Anti-infectieuses (CBSA) UR 4312, F-76000 Rouen, France"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"ORCID":"https:\/\/orcid.org\/0000-0002-9509-6054","authenticated-orcid":false,"given":"Magalie","family":"Barreau","sequence":"additional","affiliation":[{"name":"Univ Rouen Normandie, Universit\u00e9 Caen Normandie, Normandie Univ, Communication Bact\u00e9rienne et Strat\u00e9gies Anti-infectieuses (CBSA) UR 4312, F-76000 Rouen, France"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"ORCID":"https:\/\/orcid.org\/0000-0001-8235-8919","authenticated-orcid":false,"given":"Olivier","family":"Lesouhaitier","sequence":"additional","affiliation":[{"name":"Univ Rouen Normandie, Universit\u00e9 Caen Normandie, Normandie Univ, Communication Bact\u00e9rienne et Strat\u00e9gies Anti-infectieuses (CBSA) UR 4312, F-76000 Rouen, France"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"ORCID":"https:\/\/orcid.org\/0000-0001-8132-7221","authenticated-orcid":false,"given":"Michael","family":"Smietana","sequence":"additional","affiliation":[{"name":"Institut des Biomol\u00e9cules Max Mousseron, Universit\u00e9 de Montpellier, CNRS, ENSCM, 1919 route de Mende, 34095 Montpellier, France"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"ORCID":"https:\/\/orcid.org\/0000-0001-6401-0935","authenticated-orcid":false,"given":"Guillaume","family":"Clav\u00e9","sequence":"additional","affiliation":[{"name":"Institut des Biomol\u00e9cules Max Mousseron, Universit\u00e9 de Montpellier, CNRS, ENSCM, 1919 route de Mende, 34095 Montpellier, France"}],"role":[{"vocabulary":"crossref","role":"author"}]}],"member":"292","published-online":{"date-parts":[[2023]]},"reference":[{"key":"D3MD00229B\/cit1\/1","doi-asserted-by":"crossref","first-page":"476","DOI":"10.1016\/j.mib.2009.08.001","volume":"12","author":"Rice","year":"2009","journal-title":"Curr. 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