{"status":"ok","message-type":"work","message-version":"1.0.0","message":{"indexed":{"date-parts":[[2026,6,25]],"date-time":"2026-06-25T23:58:41Z","timestamp":1782431921884,"version":"3.54.5"},"reference-count":49,"publisher":"Informa UK Limited","issue":"sup2","content-domain":{"domain":["www.tandfonline.com"],"crossmark-restriction":true},"short-container-title":["Journal of Enzyme Inhibition and Medicinal Chemistry"],"published-print":{"date-parts":[[2016,11,2]]},"DOI":"10.1080\/14756366.2016.1197221","type":"journal-article","created":{"date-parts":[[2016,6,17]],"date-time":"2016-06-17T13:30:34Z","timestamp":1466170234000},"page":"174-179","update-policy":"https:\/\/doi.org\/10.1080\/tandf_crossmark_01","source":"Crossref","is-referenced-by-count":27,"title":["Design, synthesis and biological evaluation of<i>N<\/i>-(5-methyl-isoxazol-3-yl\/1,3,4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors"],"prefix":"10.1080","volume":"31","author":[{"given":"Chandra Bhushan","family":"Mishra","sequence":"first","affiliation":[{"name":"Bio-Organic Chemistry Laboratory, Dr. B. R. Ambedkar Centre for Biomedical Research, University of Delhi, Delhi, India,"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Shikha","family":"Kumari","sequence":"additional","affiliation":[{"name":"Bio-Organic Chemistry Laboratory, Dr. B. R. Ambedkar Centre for Biomedical Research, University of Delhi, Delhi, India,"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Andrea","family":"Angeli","sequence":"additional","affiliation":[{"name":"Dipartimento Neurofarba, Universit\u00e0 degli Studi di Firenze, Sezione di Scienze Farmaceutiche e Nutraceutiche, Florence, Italy,"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Simona Maria","family":"Monti","sequence":"additional","affiliation":[{"name":"Istituto di Biostrutture e Bioimmagini (IBB) CNR, via Mezzocannone, Naples, Italy, and"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Martina","family":"Buonanno","sequence":"additional","affiliation":[{"name":"Istituto di Biostrutture e Bioimmagini (IBB) CNR, via Mezzocannone, Naples, Italy, and"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Amresh","family":"Prakash","sequence":"additional","affiliation":[{"name":"School of Computational and Integrative Sciences, Jawaharlal Nehru University, New Delhi, India"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Manisha","family":"Tiwari","sequence":"additional","affiliation":[{"name":"Bio-Organic Chemistry Laboratory, Dr. B. R. Ambedkar Centre for Biomedical Research, University of Delhi, Delhi, India,"}],"role":[{"vocabulary":"crossref","role":"author"}]},{"given":"Claudiu T.","family":"Supuran","sequence":"additional","affiliation":[{"name":"Dipartimento Neurofarba, Universit\u00e0 degli Studi di Firenze, Sezione di Scienze Farmaceutiche e Nutraceutiche, Florence, Italy,"}],"role":[{"vocabulary":"crossref","role":"author"}]}],"member":"301","published-online":{"date-parts":[[2016,6,17]]},"reference":[{"key":"CIT0001","doi-asserted-by":"publisher","DOI":"10.1038\/nrd2467"},{"key":"CIT0002","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmcl.2014.08.015"},{"key":"CIT0003","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmc.2014.10.041"},{"key":"CIT0004","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2012.672983"},{"key":"CIT0005","doi-asserted-by":"publisher","DOI":"10.1021\/cr200176r"},{"key":"CIT0006","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmc.2007.04.020"},{"key":"CIT0007","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2015.1122001"},{"key":"CIT0008","doi-asserted-by":"publisher","DOI":"10.1038\/nrd3554"},{"key":"CIT0009","doi-asserted-by":"publisher","DOI":"10.4155\/fmc.14.68"},{"key":"CIT0010","first-page":"1","volume":"3","author":"Shah GN","year":"2004","journal-title":"Hum Mutat"},{"key":"CIT0011","doi-asserted-by":"publisher","DOI":"10.1002\/cmdc.200700057"},{"key":"CIT0012","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2013.761876"},{"key":"CIT0013","doi-asserted-by":"publisher","DOI":"10.1586\/14737175.2015.1066675"},{"key":"CIT0014","doi-asserted-by":"publisher","DOI":"10.1002\/med.10025"},{"key":"CIT0015","doi-asserted-by":"publisher","DOI":"10.1517\/17460441.2015.1038235"},{"key":"CIT0016","doi-asserted-by":"crossref","first-page":"2561","DOI":"10.1016\/S0021-9258(18)62326-9","volume":"246","author":"Khalifah RG.","year":"1971","journal-title":". J Biol Chem"},{"key":"CIT0017","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2011.650692"},{"key":"CIT0018","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2013.777334"},{"key":"CIT0019","doi-asserted-by":"publisher","DOI":"10.1021\/jm049692i"},{"key":"CIT0020","doi-asserted-by":"publisher","DOI":"10.1021\/jm001051+"},{"key":"CIT0021","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmcl.2005.06.054"},{"key":"CIT0022","doi-asserted-by":"publisher","DOI":"10.1016\/S0223-5234(98)80033-0"},{"key":"CIT0023","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmcl.2010.06.082"},{"key":"CIT0024","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmc.2010.06.028"},{"key":"CIT0025","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmc.2011.04.005"},{"key":"CIT0026","doi-asserted-by":"publisher","DOI":"10.1021\/jm200209n"},{"key":"CIT0027","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmc.2013.02.022"},{"key":"CIT0028","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmcl.2005.01.086"},{"key":"CIT0029","doi-asserted-by":"publisher","DOI":"10.1021\/jm900641r"},{"key":"CIT0030","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmcl.2007.12.022"},{"key":"CIT0031","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmcl.2005.03.032"},{"key":"CIT0032","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmcl.2011.12.134"},{"key":"CIT0033","doi-asserted-by":"publisher","DOI":"10.1158\/0008-5472.CAN-10-4261"},{"key":"CIT0034","doi-asserted-by":"publisher","DOI":"10.1021\/jm101541x"},{"key":"CIT0035","doi-asserted-by":"publisher","DOI":"10.1517\/13543776.2013.742065"},{"key":"CIT0036","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2011.617745"},{"key":"CIT0037","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2012.732071"},{"key":"CIT0038","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2014.880696"},{"key":"CIT0039","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2014.983917"},{"key":"CIT0040","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2011.638921"},{"key":"CIT0041","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmc.2012.05.037"},{"key":"CIT0042","doi-asserted-by":"publisher","DOI":"10.1039\/c3cc40858b"},{"key":"CIT0043","doi-asserted-by":"publisher","DOI":"10.3109\/14756366.2014.963072"},{"key":"CIT0044","doi-asserted-by":"crossref","first-page":"1821","DOI":"10.1016\/j.bmc.2014.01.056","volume":"22","author":"D'Ascenzio M","year":"2014","journal-title":"Bioorg Med Chem"},{"key":"CIT0045","doi-asserted-by":"publisher","DOI":"10.1016\/j.ejmech.2014.07.014"},{"key":"CIT0046","doi-asserted-by":"crossref","first-page":"3982","DOI":"10.1016\/j.bmc.2014.06.003","volume":"22","author":"D'Ascenzio M","year":"2014","journal-title":"Bioorg Med Chem"},{"key":"CIT0047","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmc.2015.05.013"},{"key":"CIT0048","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmc.2015.07.066"},{"key":"CIT0049","doi-asserted-by":"publisher","DOI":"10.1016\/j.bmc.2012.10.048"}],"container-title":["Journal of Enzyme Inhibition and Medicinal Chemistry"],"original-title":[],"language":"en","link":[{"URL":"https:\/\/www.tandfonline.com\/doi\/pdf\/10.1080\/14756366.2016.1197221","content-type":"unspecified","content-version":"vor","intended-application":"similarity-checking"}],"deposited":{"date-parts":[[2022,7,1]],"date-time":"2022-07-01T21:50:13Z","timestamp":1656712213000},"score":1,"resource":{"primary":{"URL":"https:\/\/www.tandfonline.com\/doi\/full\/10.1080\/14756366.2016.1197221"}},"subtitle":[],"short-title":[],"issued":{"date-parts":[[2016,6,17]]},"references-count":49,"journal-issue":{"issue":"sup2","published-print":{"date-parts":[[2016,11,2]]}},"alternative-id":["10.1080\/14756366.2016.1197221"],"URL":"https:\/\/doi.org\/10.1080\/14756366.2016.1197221","relation":{},"ISSN":["1475-6366","1475-6374"],"issn-type":[{"value":"1475-6366","type":"print"},{"value":"1475-6374","type":"electronic"}],"subject":[],"published":{"date-parts":[[2016,6,17]]},"assertion":[{"value":"The publishing and review policy for this title is described in its Aims & Scope.","order":1,"name":"peerreview_statement","label":"Peer Review Statement"},{"value":"http:\/\/www.tandfonline.com\/action\/journalInformation?show=aimsScope&journalCode=ienz20","URL":"http:\/\/www.tandfonline.com\/action\/journalInformation?show=aimsScope&journalCode=ienz20","order":2,"name":"aims_and_scope_url","label":"Aim & Scope"},{"value":"2016-05-16","order":0,"name":"received","label":"Received","group":{"name":"publication_history","label":"Publication History"}},{"value":"2016-05-31","order":2,"name":"accepted","label":"Accepted","group":{"name":"publication_history","label":"Publication History"}},{"value":"2016-06-17","order":3,"name":"published","label":"Published","group":{"name":"publication_history","label":"Publication History"}}]}}