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Med. Biol."],"published-print":{"date-parts":[[2026,10,28]]},"abstract":"<jats:title>Abstract<\/jats:title>\n                  <jats:p>\n                    <jats:italic>Objective<\/jats:italic>\n                    . Tellurium-118 (\n                    <jats:sup>118<\/jats:sup>\n                    Te;\n                    <jats:italic>t<\/jats:italic>\n                    <jats:sub>1\/2<\/jats:sub>\n                    = 6.00 \u00b1 0.02 d) can act as an\n                    <jats:italic>in vivo<\/jats:italic>\n                    generator of the positron emitter antimony-118 (\n                    <jats:sup>118<\/jats:sup>\n                    Sb;\n                    <jats:italic>t<\/jats:italic>\n                    <jats:sub>1\/2<\/jats:sub>\n                    = 3.6 \u00b1 0.3 min), enabling positron emission tomography (PET) over a week or longer. This work assessed absorbed doses associated with free\n                    <jats:sup>118<\/jats:sup>\n                    Te to establish a dosimetric safety basis for\n                    <jats:sup>118<\/jats:sup>\n                    Te radiopharmaceuticals.\n                    <jats:italic>Approach<\/jats:italic>\n                    . Injection solutions of free\n                    <jats:sup>118<\/jats:sup>\n                    Te were prepared by alpha-particle irradiation of an enriched tin-116 target followed by radiochemical isolation.\n                    <jats:italic>Ex vivo<\/jats:italic>\n                    biodistribution in healthy female Slc:ICR mice was acquired at seven time points from 2 h to 29 d postinjection (\n                    <jats:italic>n<\/jats:italic>\n                    = 6 per time point). Time-integrated activity coefficients were computed from the biodistribution profiles and extrapolated to a human model using relative mass scaling. Absorbed dose coefficients (ADCs) were calculated following the medical internal radiation dose formalism with computational phantoms implemented in the dosimetry software OLINDA. Dosimetric contributions from\n                    <jats:sup>118<\/jats:sup>\n                    Te and its coproduced radioisotopic impurity\n                    <jats:sup>119m<\/jats:sup>\n                    Te (\n                    <jats:italic>t<\/jats:italic>\n                    <jats:sub>1\/2<\/jats:sub>\n                    = 4.69 \u00b1 0.04 d), along with their equilibrium daughters\n                    <jats:sup>118<\/jats:sup>\n                    Sb and\n                    <jats:sup>119<\/jats:sup>\n                    Sb, were individually assessed.\n                    <jats:italic>Main results<\/jats:italic>\n                    . The kidneys exhibited the highest ADC in both mouse (2666.0 mGy MBq\n                    <jats:sup>\u22121<\/jats:sup>\n                    ) and human (2.639 mGy MBq\n                    <jats:sup>\u22121<\/jats:sup>\n                    ) models. Bone received the second-highest ADC in the mouse model, 1855.5 mGy MBq\n                    <jats:sup>\u22121<\/jats:sup>\n                    . Antimony-118 dominated absorbed doses across all organs examined, accounting for more than 82% of ADCs in both models. Contributions from\n                    <jats:sup>118<\/jats:sup>\n                    Te,\n                    <jats:sup>119m<\/jats:sup>\n                    Te, and\n                    <jats:sup>119<\/jats:sup>\n                    Sb were minor by comparison.\n                    <jats:italic>Significance<\/jats:italic>\n                    . The kidneys and bone were identified as the primary dosimetric targets of free\n                    <jats:sup>118<\/jats:sup>\n                    Te, with its daughter\n                    <jats:sup>118<\/jats:sup>\n                    Sb being the principal dose contributor. The limited dosimetric impact from\n                    <jats:sup>118<\/jats:sup>\n                    Te provides justification for its use as an\n                    <jats:italic>in vivo<\/jats:italic>\n                    generator of\n                    <jats:sup>118<\/jats:sup>\n                    Sb for long-term PET. The ADCs reported here offer a quantitative basis for assessing the dosimetric safety of\n                    <jats:sup>118<\/jats:sup>\n                    Te radiopharmaceuticals.\n                  <\/jats:p>","DOI":"10.1088\/1361-6560\/aeb089","type":"journal-article","created":{"date-parts":[[2026,10,5]],"date-time":"2026-10-05T22:54:37Z","timestamp":1791240877000},"page":"205036","update-policy":"https:\/\/doi.org\/10.1088\/crossmark-policy","source":"Crossref","is-referenced-by-count":0,"title":["Biodistribution and dosimetry of free\n                    <sup>118<\/sup>\n                    Te, an\n                    <i>in vivo<\/i>\n                    generator of the positron emitter\n                    <sup>118<\/sup>\n                    Sb for long-term positron emission 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All rights, including for text and data mining, AI training, and similar technologies, are reserved.","name":"copyright_information","label":"Copyright Information"},{"value":"2026-06-10","name":"date_received","label":"Date Received","group":{"name":"publication_dates","label":"Publication dates"}},{"value":"2026-10-05","name":"date_accepted","label":"Date Accepted","group":{"name":"publication_dates","label":"Publication dates"}},{"value":"2026-10-28","name":"date_epub","label":"Online publication date","group":{"name":"publication_dates","label":"Publication dates"}}]}}