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The worldwide known antidiabetic use of the drug has been suggested to arise from a complex combination effect of various constituents. Moreover, the drug is also a potential antihyperuricemic agent. Considering that type 2 diabetes and hyperuricemia are vice-versa in each other\u2019s important risk factors, the use of mulberry originated phytotherapeutics might provide an excellent option for the prevention and\/or treatment of both conditions. Here we report a series of relevant<jats:italic>in vitro<\/jats:italic>and<jats:italic>in vivo<\/jats:italic>studies on the bioactivity of an extract of mulberry leaves and its fractions obtained by a stepwise gradient on silica gel.<jats:italic>In vivo<\/jats:italic>antihyperglycemic and antihyperuricemic activity, plasma antioxidant status, as well as<jats:italic>in vitro<\/jats:italic>glucose consumption by adipocytes in the presence or absence of insulin, xanthine oxidase inhibition, free radical scavenging activity, and inhibition of lipid peroxidation were tested. Known bioactive constituents of<jats:italic>M. alba<\/jats:italic>(chlorogenic acid, rutin, isoquercitrin, and loliolide) were identified and quantified from the HPLC-DAD fingerprint chromatograms. Iminosugar contents were investigated by MS\/MS, 1-deoxynojirimycin was quantified, and amounts of 2-<jats:italic>O<\/jats:italic>-alpha-D-galactopyranosyl-1-deoxynojirimicin and fagomine were additionally estimated.<\/jats:p>","DOI":"10.1155\/2013\/948627","type":"journal-article","created":{"date-parts":[[2013,12,5]],"date-time":"2013-12-05T21:15:53Z","timestamp":1386278153000},"page":"1-10","source":"Crossref","is-referenced-by-count":34,"title":["Metabolic Effects of Mulberry Leaves: Exploring Potential Benefits in Type 2 Diabetes and Hyperuricemia"],"prefix":"10.1155","volume":"2013","author":[{"given":"A.","family":"Hunyadi","sequence":"first","affiliation":[{"name":"Institute of Pharmacognosy, Faculty of Pharmacy, University of Szeged, E\u00f6tv\u00f6s u. 6, Szeged 6720, Hungary"}]},{"given":"E.","family":"Liktor-Busa","sequence":"additional","affiliation":[{"name":"Institute of Pharmacognosy, Faculty of Pharmacy, University of Szeged, E\u00f6tv\u00f6s u. 6, Szeged 6720, Hungary"}]},{"given":"\u00c1.","family":"M\u00e1rki","sequence":"additional","affiliation":[{"name":"Department of Pharmacodynamics and Biopharmacy, Faculty of Pharmacy, University of Szeged, E\u00f6tv\u00f6s u. 6, Szeged 6720, Hungary"}]},{"given":"A.","family":"Martins","sequence":"additional","affiliation":[{"name":"Department of Medical Microbiology and Immunobiology, Faculty of Medicine, University of Szeged, D\u00f3m t\u00e9r 13, Szeged 6720, Hungary"},{"name":"Unidade de Parasitologia e Microbiologia M\u00e9dica, Instituto de Higiene e Medicina Tropical, Universidade Nova de Lisboa, Rua da Junqueira 100, 1349-008 Lisboa, Portugal"}]},{"given":"N.","family":"Jedlinszki","sequence":"additional","affiliation":[{"name":"Institute of Pharmacognosy, Faculty of Pharmacy, University of Szeged, E\u00f6tv\u00f6s u. 6, Szeged 6720, Hungary"}]},{"given":"T. J.","family":"Hsieh","sequence":"additional","affiliation":[{"name":"Department of Genome Medicine, College of Medicine, Kaohsiung Medical University, Shih Chuan 1st Rd. 100, Kaohsiung 807, Taiwan"}]},{"given":"M.","family":"B\u00e1thori","sequence":"additional","affiliation":[{"name":"Institute of Pharmacognosy, Faculty of Pharmacy, University of Szeged, E\u00f6tv\u00f6s u. 6, Szeged 6720, Hungary"}]},{"given":"J.","family":"Hohmann","sequence":"additional","affiliation":[{"name":"Institute of Pharmacognosy, Faculty of Pharmacy, University of Szeged, E\u00f6tv\u00f6s u. 6, Szeged 6720, Hungary"}]},{"given":"I.","family":"Zupk\u00f3","sequence":"additional","affiliation":[{"name":"Department of Pharmacodynamics and Biopharmacy, Faculty of Pharmacy, University of Szeged, E\u00f6tv\u00f6s u. 6, Szeged 6720, 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