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Ministry of Health, Labour and Welfare (2011)."},{"key":"3","unstructured":"3) Japan College of Rheumatology. <i>Rheumatology Disease Text Revision<\/i>, 2nd Ed., Shindan to Chiryo Sha, Inc., Tokyo, pp. 7\u201359 (2016)."},{"key":"4","unstructured":"4) Sugawara T. <i>New product development and clinical needs for bone joint cartilage treatment<\/i>. Technical Information Institute Co., Ltd., pp. 22\u201327, 237\u2013241 (2015)."},{"key":"5","unstructured":"5) Pfizer Inc. Rumatrex capsule 2\u2009mg Interview Form Revised February 19th edition (2016)."},{"key":"6","unstructured":"6) AbbVie Inc. Humira subcutaneous injection formulation Interview Form 15th ed. (2016)."},{"key":"7","doi-asserted-by":"crossref","unstructured":"7) Okuda T, Kobayashi Y, Yanamoto S, Okamoto H. PEG conjugation of a near-infrared fluorescent probe for noninvasive dual imaging of lung deposition and gene expression by pulmonary gene delivery. <i>J. 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J.<\/i> <i>Joint Diseases<\/i>, <b>33<\/b>, 19\u201324 (2014)."},{"key":"12","doi-asserted-by":"crossref","unstructured":"12) Gotoh S, Miyazaki K, Onaya J, Sakamoto T, Tokuyasu K, Namiki O. Experimental knee pain model in rats and analgesic effect of sodium hyaluronate (SPH). <i>Nippon Yakurigaku Zasshi<\/i>, <b>92<\/b>, 17\u201327 (1988).","DOI":"10.1254\/fpj.92.17"},{"key":"13","unstructured":"13) Yamashita I, Atsuta Y, Shimazaki S, Miyatsu M. Effects of prostaglandin E2 and sodium hyaluronate on bradykinin induced knee joint pain in rat. <i>Nihon Seikeigeka Gakkai Zasshi<\/i>, <b>69<\/b>, 735\u2013743 (1995)."},{"key":"14","doi-asserted-by":"crossref","unstructured":"14) Aihara S, Murakami T, Ishii R, Tempo R, Higashi Y, Hamada K, Umemoto K, Maeda S. Effect of sodium hyaluronate on experimental arthritic pain in rats. <i>Maeda Jap. Pharmacol. J.<\/i>, <b>100<\/b>, 359\u2013365 (1992).","DOI":"10.1254\/fpj.100.359"},{"key":"15","unstructured":"15) Tsuruhara Pharmaceutical Co., Ltd. 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Prolonged anti-inflammatory action of DL-lactide\/glycolide copolymer nanospheres containing betamethasone sodium phosphate for an intra-articular delivery system in antigen-induced arthritic rabbit. <i>Pharm. Res.<\/i>, <b>19<\/b>, 403\u2013410 (2002).","DOI":"10.1023\/A:1015123024113"},{"key":"19","doi-asserted-by":"crossref","unstructured":"19) Horisawa E, Kubota K, Tuboi I, Sato K, Yamamoto H, Takeuchi H, Kawashima Y. Size-dependency of DL-lactide\/glycolide copolymer particulates for intra-articular delivery system on phagocytosis in rat synovium. <i>Pharm. Res.<\/i>, <b>19<\/b>, 132\u2013139 (2002).","DOI":"10.1023\/A:1014260513728"},{"key":"20","doi-asserted-by":"crossref","unstructured":"20) Kim SR, Ho MJ, Lee E, Lee JW, Choi YW, Kang MJ. Cationic PLGA\/Eudragit RL nanoparticles for increasing retention time in synovial cavity after intra-articular injection in knee joint. <i>Int. J. 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