none 10.3987/COM-99-8635 CLOCKSS Archive CLOCKSS Archive 5187 36606090 73640 20090312102723 10.13030 2024-06-24T20:52:47Z 2009-03-12T02:57:44Z 16 HETEROCYCLES HETEROCYCLES 0385-5414 HTCYAM 1999 51 10 Synthesis of Trifluoromethylpyrimidines from Fluorinated En-aminodiketones Catherine Mirand Mustapha Soufyane Sarah van den Broek Layachi Khamliche 1999 2445 COM-99-8635 10.3987/COM-99-8635 20090312102723 https://triggered.stanford.clockss.org/ServeContent?doi=10.3987%2Fcom-99-8635 https://triggered.edinburgh.clockss.org/ServeContent?doi=10.3987%2Fcom-99-8635 10.1016/S0040-4039(00)93433-6 1. J. Lévy, M. Soufyane, C. Mirand, M. Döé de Maindreville, and D. Royer, Tetrahedron Lett., 1991, 32, 5081. 10.1016/S0040-4039(00)61552-6 2. M. Soufyane, C. Mirand, and J. Lévy, Tetrahedron Lett., 1993, 34, 7737. 3. A new synthesis of DAMFA was recently described by A. V. Sanin, V. G. Nenajdenko, K. I. Smolko, D. I. Denisenko, and E. S. Balenkova, Synthesis, 1998, 842. a) R. Filler and Y. Kobayashi, ‘Biomedicinal Aspects of Fluorine Chemistry’, Kodansha & Elsevier Biomedical, New York, 1982; 10.1016/S0040-4020(01)90286-8 b) J. T. Welch, Tetrahedron, 1987, 43, 3123. 10.1021/jm9508649 a) P. Dorigo, D. Fraccarollo, G. Santostasi, I. Maragno, M. Floreani, P. A. Borea, L. Mosti, L. Sansebastiano, P. Fossa, F. Orsini, F. Benetello, and G. Bombieri, J. Med. Chem., 1996, 39, 3671; 10.1016/0040-4039(96)00129-3 b) H. Yamanaka, T. Takekawa, K. Morita, T. Ishihara, and J. T. Gupton, Tetrahedron Lett., 1996, 37, 1829; 10.3987/COM-96-S26 c) E. Okada, T. Kinomura, H. Takeuchi, and M. Hojo, Heterocycles, 1997, 44, 349; 10.1016/S0040-4039(96)02256-3 d) L. M. Gayo and M. J. Suto, Tetrahedron Lett., 1997, 38, 211; 10.1055/s-1997-1376 e) H. P. Guan, X. Q. Tang, B. H. Luo, and C. M. Hu, Synthesis, 1997, 1489. 10.1021/jo01016a012 6. W. J. Middleton and C. G. Krespan, J. Org. Chem., 1965, 30, 1398. 10.1016/0040-4020(79)88001-1 a) R. F. Abdulla and R. S. Brinkmeyer, Tetrahedron, 1979, 35, 1675; 10.1002/jlac.19616410102 b) H. Meerwein, W. Florian, N. Schön, and G. Stopp, Liebigs Ann., 1961, 641, 1. 10.1021/jo00138a033 8. W. Verboom, D. N. Reinhouldt, S. Harkema, and G. J. Van Hummel, J. Org. Chem., 1982, 47, 3339.